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N-[4-(furan-2-yl)butan-2-yl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
({4-ethyl-5-[1-(2-ethylpyrimidine-5-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
2-({2-amino-6-[2-(aminomethyl)-4-fluoro-2,3-dihydro-1-benzofuran-7-yl]pyrimidin-4-yl}amino)ethan-1-ol
6-[3-(hydroxymethyl)pyrrolidin-1-yl]-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
2-[(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)amino]pyridine-3-carboxamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-methoxypyridine-3-carboxamide
N,2,6-trimethyl-N-(quinoxalin-6-ylmethyl)quinoline-4-carboxamide
4-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]-N-(4-methylphenyl)piperidine-1-carboxamide
3-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]-1-(1,2,3,4-tetrahydroquinolin-1-yl)propan-1-one
2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
4-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholine-4-carbonyl)pyridin-2-amine
N,N-diethyl-4-(3-methylpyridin-4-yl)benzamide
1-cyclopropyl-N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-5-oxopyrrolidine-3-carboxamide
2-(2-fluorophenyl)-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)acetamide
1-(3-methylpyridin-4-yl)-4-(2,2,6,6-tetramethylpiperidin-4-yl)-1,4-diazepane
4-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]-1-ethyl-1,2-dihydropyridin-2-one
4,6-dimethyl-1-(2-{[1-(9H-purin-6-yl)piperidin-4-yl]amino}ethyl)-1,2-dihydropyrimidin-2-one
3-{[4-(cyclobutylmethyl)piperazin-1-yl]methyl}-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one
7-(3-chlorophenyl)-4-[(4-hydroxy-3-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(2R,3R)-3-(dimethylamino)-1'-(3-fluoropyridine-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-(1-ethyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-[(2-fluorophenyl)methyl]piperazin-2-one
7-(1,3-benzothiazol-2-yl)-4-(2,2-difluorocyclopropanecarbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-methyl-N-{[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-3-yl]methyl}-1,2-oxazole-3-carboxamide
7-chloro-4-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-1λ6-thiomorpholine-1,1-dione
N-[(2R,3R)-2-methoxy-1'-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
5-acetyl-2,4-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1H-pyrrole-3-carboxamide
6-chloro-N,N-dimethyl-3-[({[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amino)methyl]imidazo[1,2-a]pyridine-2-carboxamide
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-(morpholin-4-yl)benzamide
(2R,6S)-2,6-dimethyl-4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)morpholine
3-(isoquinolin-1-yl)benzonitrile
N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-(trifluoromethyl)benzamide
N-[2-(cyclohexylsulfanyl)ethyl]-6-(methoxymethyl)pyrimidin-4-amine
4-({2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)benzonitrile
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
N-{1-[7-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}acetamide
2-{1-[(2E)-3-phenylprop-2-en-1-yl]azetidin-3-yl}pyridine
5-tert-butyl-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1,3,4-oxadiazol-2-amine
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methylpiperazine
1-cyclopentyl-N-[3-(3-methyl-1H-pyrazol-1-yl)propyl]-5-oxopyrrolidine-3-carboxamide
6-methyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}imidazo[2,1-b][1,3]thiazole-5-carboxamide
7-cyclopentyl-2-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(2-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
1-[(4-fluorophenyl)methyl]-4-{2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}piperazin-2-one
2-methyl-4-(pyridin-4-yl)quinazoline
3-(2,5-difluorobenzoyl)-1-[(2,3,4-trimethoxyphenyl)methyl]piperidine
methyl 2-hydroxy-5-[(2-methyl-5-oxo-1,4-diazepan-1-yl)methyl]benzoate
1-phenyl-4-[2-(2-phenylethyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
5-(2,4-dimethoxyphenyl)-N-[1-(6-methylpyridin-2-yl)propan-2-yl]-1,2,4-triazin-3-amine