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N-benzyl-N-(3-hydroxy-2-methylpropyl)-4-(hydroxymethyl)benzamide
N-[(5-chlorothiophen-2-yl)methyl]-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-[4-({3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1,2-oxazol-5-yl}methoxy)-3-methoxyphenyl]ethan-1-one
N-[(3S,4R)-1-[(2,3-dimethyl-1H-indol-7-yl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
5-[1-(furan-2-ylmethyl)pyrrolidin-2-yl]-N-(trimethyl-1H-pyrazol-4-yl)thiophene-2-carboxamide
[3-(2-methoxyethyl)-1-(1H-pyrrole-3-carbonyl)piperidin-3-yl]methanol
N,2,3,5-tetramethyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
8-acetyl-2-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(3aR,7aS)-2-(5-methanesulfonyl-2-methylpyrimidin-4-yl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-(oxolan-2-ylmethyl)-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
3-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1-{4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]phenyl}urea
6-chloro-8-methyl-3-(1H-1,2,3,4-tetrazol-5-ylmethyl)-3,4-dihydroquinazolin-4-one
5-(1H-indol-1-ylmethyl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}furan-2-carboxamide
1-(carbamoylmethyl)-N-[2-(2-ethoxyphenoxy)ethyl]-N-methylpiperidine-4-carboxamide
2-methoxy-N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)acetamide
(1-benzothiophen-2-ylmethyl)({[4-({1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-4-yl}oxy)phenyl]methyl})methylamine
2-{1-[5-(naphthalen-2-yl)-1,2,4-triazin-3-yl]piperidin-4-yl}-1H-1,3-benzodiazole
4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[2-(1-methylpiperidin-3-yl)ethyl]benzamide
ethyl 3-benzyl-1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidine-3-carboxylate
3-methyl-1-[(4-methylphenyl)methyl]-4-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-2-one
2-(methylsulfanyl)-1-{3-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidin-1-yl}ethan-1-one
7-(1-benzothiophen-3-yl)-4-(5-methyl-1,2-oxazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(3,4-difluorophenyl)-3-methyl-5-[2-(1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazole
ethyl 4-[(4-chlorophenyl)methyl]-1-[(2-hydroxyphenyl)methyl]piperidine-4-carboxylate
1-[(5-ethylpyridin-2-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
2-(but-3-enoyl)-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
5-(2H-1,3-benzodioxol-5-yl)-1-ethyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
methyl 3-(2-cyclopentylacetamido)-6-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
5-(1-cyclopentanecarbonylpiperidin-4-yl)-3-[3-(dimethylamino)propyl]-5-[(4-fluorophenyl)methyl]imidazolidine-2,4-dione
(1R,5R)-6-(2-methoxyethyl)-3-[2-(methylsulfanyl)pyridine-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(3aR,6aR)-2-{[4-(methylsulfanyl)phenyl]methyl}-5-(pyridin-3-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-cyclopropyl-7-{imidazo[1,2-a]pyridine-3-carbonyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(4-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-N,N-dimethylacetamide
1-(1,5-dimethyl-1H-pyrazol-4-yl)-3-[2-(dimethylsulfamoyl)ethyl]urea
N-[2-(2-methoxyphenyl)ethyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-[2-methyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-4-(pyrimidin-2-yloxy)piperidine-1-carboxamide
4-(4-chlorophenyl)-N-ethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]butanamide
(2S,4S)-4-amino-N-ethyl-1-[3-(1H-pyrazol-4-yl)benzoyl]pyrrolidine-2-carboxamide
4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}thiomorpholine
1-(2-chlorophenyl)-3-{1-[1-(2-oxo-2-phenylacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
5-[(3-hydroxyazetidin-1-yl)methyl]-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-N,1,4,6-tetramethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-[5-(furan-2-yl)-1,3,4-thiadiazol-2-yl]-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)urea
2-{[3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazin-1-yl]methyl}-3-methoxyphenol
{1-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
N-(1-benzofuran-2-ylmethyl)-1-(pyrimidin-2-yl)piperidin-3-amine
5-ethyl-N-{[3-methyl-7-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1,2-oxazole-3-carboxamide
4-[(5-chloro-2,3-dimethoxyphenyl)methyl]morpholine
N-{1-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide