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4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[(2S)-oxolan-2-ylmethyl]benzamide
ethyl 4-{2-[1-benzyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetyl}piperazine-1-carboxylate
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-methyl-1-[(3-methylphenyl)methyl]pyrrolidine-2-carboxamide
N-ethyl-8-methoxy-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-{4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidine-1-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
10-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
5-[5-(2,3-dihydro-1-benzofuran-5-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
3-(2-ethyl-1H-imidazol-1-yl)-1-[3-(4-phenoxybenzoyl)piperidin-1-yl]propan-1-one
3-[2-(trifluoromethyl)morpholine-4-carbonyl]pyridin-2-ol
5-[({1-[3-(1,3-thiazol-4-yl)phenyl]piperidin-4-yl}amino)methyl]pyrrolidin-2-one
4-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decane-7-carbonyl}benzonitrile
N-(2-hydroxy-2-phenylethyl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
2-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-5-methylpyrazine
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]pyrrolidine-1-sulfonamide
3-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
2-(4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1-(2,2-dimethylpropyl)piperazin-2-yl)ethan-1-ol
methyl (2S,4R)-4-(dimethylamino)-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]pyrrolidine-2-carboxylate
4-{2-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-oxoethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
N-methyl-4-(piperidin-3-yl)-N-(quinolin-3-ylmethyl)benzamide
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-3-[(3-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N,N-dimethyl-3-({2-[(3-methylpyridin-2-yl)amino]ethyl}sulfamoyl)benzamide
3-(2-chlorophenyl)-6-(5-ethyl-1,2-oxazole-3-carbonyl)-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(1R,3s,6r,8S)-4-[5-(2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-azatricyclo[4.3.1.13,8]undecane
1-[(2E)-3-phenylprop-2-en-1-yl]-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
4-(3-phenylpropyl)-1-(pyridin-2-ylmethyl)piperidine-4-carboxylic acid
1-(2,3-dihydro-1H-inden-2-yl)-4-({[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}amino)pyrrolidin-2-one
1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-methylpiperazine
1-{6-[({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]pyridin-3-yl}ethan-1-one
1-[2-(dimethylamino)ethyl]-3-(3-fluorophenyl)-3-{2-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2,3-dihydro-1H-indene-1-carboxamide
1-cyclopropyl-5-oxo-N-[2-(3-phenoxyphenyl)ethyl]pyrrolidine-3-carboxamide
1-{1-[(5-phenylthiophen-2-yl)methyl]piperidin-3-yl}pyrrolidin-2-one
4-chloro-2-hydroxy-N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}benzamide
N-methyl-3-(1,2-oxazinan-2-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
N-[2-(2-{8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-2-oxoacetyl)phenyl]propanamide
methyl 3-(2,6-dimethoxybenzoyl)-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[2-(1H-pyrazol-1-yl)ethyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(2,5-difluorophenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
2-{1-[(3-methoxyphenyl)methyl]-4-(1H-pyrazol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
1-[9-(but-3-yn-1-yloxy)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
4-[(3R,4S)-3-(1-methyl-2-oxo-1,2-dihydropyridine-3-amido)-4-(propan-2-yl)pyrrolidin-1-yl]butanoic acid
1-[(4-chlorophenyl)methyl]-4-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperazine
7-(3-chlorophenyl)-4-(2-methylbenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-(5-methylthiophen-2-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-(3-methoxy-5-methylthiophene-2-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
5-(3-methoxyphenyl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1,2,4-triazin-3-amine
6-[2-({2-amino-6-[(4-fluorophenyl)sulfanyl]pyrimidin-4-yl}amino)ethyl]-3,4-dihydropyrimidin-4-one
(3aS,6aS)-2-(ethanesulfonyl)-5-(5-methylthiophene-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-methyl-1-(3-phenylbutyl)-1,4-diazepan-5-one
[(2S,6S)-4-[4-(morpholin-4-yl)benzoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol