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4-[4-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperazin-1-yl]-6-ethylpyrimidine
3-(2-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
3-{[1-(1,2,4-oxadiazol-3-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
9-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 2-{[6-(4-chlorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}-4-(methylsulfanyl)butanoate
1-(3,4-dichlorophenyl)-4-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]piperazine
methyl 1-[3-(4-{[ethyl(methyl)amino]methyl}phenoxy)-2-hydroxypropyl]piperidine-4-carboxylate
2-(2-{[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]methyl}phenoxy)acetic acid
1-acetyl-N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]piperidine-3-carboxamide
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-3-(methylsulfanyl)propanamide
1-(2-fluorophenyl)-N-[1-(methoxymethyl)cyclopentyl]-2,2-dimethylcyclopropane-1-carboxamide
N-[(3-chloro-1-benzothiophen-2-yl)methyl]-N-methyl-2-(methylamino)acetamide
4-{4-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]piperazin-1-yl}-2-methyl-6-propylpyrimidine
N-ethyl-2-{8-methyl-3-oxo-2,8-diazaspiro[4.5]decan-2-yl}-N-[(5-methylfuran-2-yl)methyl]acetamide
N-[2-(azepan-1-yl)ethyl]-N-ethyl-2-(morpholin-2-yl)acetamide
ethyl 2-{2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}propanoate
1-benzyl-N,2-dimethyl-5-(2-methylpropanamido)-N-(thiophen-3-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
N-[4-(azepan-1-yl)butyl]-5-hydroxypyridine-2-carboxamide
N-[2-(diethylamino)ethyl]-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-ethyl-5-methyl-1H-pyrazole-4-carboxamide
2-(3-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)-N-propylaniline
2-{2-[4-(trifluoromethyl)phenyl]-1H-imidazol-1-yl}ethan-1-ol
1-(furan-2-carbonyl)-4-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)-1,4-diazepane
2-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-N-(1,3-thiazol-2-yl)butanamide
(2S)-2-amino-N-methyl-2-phenyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
4-[5-(propan-2-yl)pyrimidin-4-yl]-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
4-cyclobutyl-6-methyl-N-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}pyrimidin-2-amine
7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-4-(4-methylpiperazine-1-carbonyl)quinoline
5-(3-fluorophenoxymethyl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]-N-(thiophen-3-ylmethyl)propanamide
(2S,4S)-N-(1-benzothiophen-2-ylmethyl)-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-1-[(4-methoxynaphthalen-1-yl)methyl]-N-methylpyrrolidine-2-carboxamide
2,6-dihydroxy-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}benzamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
3-[({1-[(2-chloro-6-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)(methyl)amino]-1λ6-thiolane-1,1-dione
1-[(2-aminopyrimidin-5-yl)methyl]-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide
N-[(3R,5S)-1-acetyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
ethyl 1-(prop-2-en-1-yl)-5-(pyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
1-(4-ethyl-1,4-diazepan-1-yl)-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
3-(1-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-4-phenyl-1H-imidazol-5-yl)phenol
3-[(4-methoxyphenyl)methyl]-1,8-bis(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
1-[5-(4-chlorophenyl)-4-methyl-1H-pyrazole-3-carbonyl]azepan-3-amine
8-(1,2,3,4-tetrahydroisoquinolin-5-yl)quinolin-4-amine
2,6-dimethyl-8-[(thiolan-3-yl)amino]octan-2-ol
2-(1H-imidazol-4-yl)-1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]ethan-1-one
2-[4-(5-{[(2-methylphenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidin-1-yl]propanamide
2-{4-[(5-methylfuran-2-yl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amine
4-{1-[(2,6-difluorophenyl)methyl]piperidin-3-yl}-5-(4-fluorophenyl)-2-methylpyrimidine
N-[(3,5-difluorophenyl)methyl]-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine