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4-methyl-2-{2-[(5-phenyl-1,2-oxazol-3-yl)formamido]ethyl}-1,3-thiazole-5-carboxylic acid
methyl 7-oxo-9-(thiophen-3-ylmethoxy)-3-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[3-({[3-(dimethyl-1,3-thiazol-2-yl)propyl]carbamoyl}amino)phenyl]-N,N-dimethylacetamide
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl){[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
N-[(1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}pyrrolidin-3-yl)methyl]but-3-enamide
[(5-chlorofuran-2-yl)methyl](methyl)[(1-methylpiperidin-3-yl)methyl]amine
methyl (2S)-1-[2-(4-{4-[(oxan-4-yl)amino]piperidin-1-yl}phenyl)acetyl]pyrrolidine-2-carboxylate
N-{[3-(4-methanesulfonylphenyl)-4-methoxyphenyl]methyl}cyclopentanamine
N-{1-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-1-oxopropan-2-yl}methanesulfonamide
2-amino-N-(1-cycloheptylpiperidin-3-yl)-6-methylpyrimidine-4-carboxamide
(oxolan-2-ylmethyl)({[5-(1H-pyrazol-5-yl)furan-2-yl]methyl})(pyridin-2-ylmethyl)amine
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-2-(trifluoromethyl)morpholine
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-3,5,7-trimethyl-1H-indole
7-chloro-N,3,5-trimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-benzofuran-2-carboxamide
3-[6-(cyclopropylamino)pyridazin-3-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
1-ethyl-4-{3-[(1-methylpiperidin-4-yl)methyl]-1-phenyl-1H-1,2,4-triazol-5-yl}-1,2-dihydropyridin-2-one
[(2S)-1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl]methanol
4-[(dimethyl-1,2-oxazol-4-yl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
8-(furan-2-ylmethyl)-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(3,4-dimethoxyphenyl)methyl]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,3-benzoxazole-6-carboxamide
3-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-3-yl]-N-(4-fluoro-2-methylphenyl)propanamide
5-[2-(2-ethoxyphenyl)-1H-imidazol-1-yl]-6-methoxy-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-(5-{[(dimethylcarbamoyl)amino]methyl}-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl)acetic acid
2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-(3-hydroxyphenyl)pyridine-3-carbonitrile
3-{[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl](methyl)amino}propan-1-ol
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-5-ethylimidazolidine-2,4-dione
(4aR,8aS)-1-(2H-1,3-benzodioxol-5-ylmethyl)-6-(4-methylbenzoyl)-decahydro-1,6-naphthyridin-2-one
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]thiophene-2-carboxamide
5-fluoro-2-{3-[4-(pyrazin-2-yl)piperazin-1-yl]propyl}-1H-1,3-benzodiazole
1-[(2-butyl-1H-imidazol-4-yl)methyl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
3-{[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}-4H-chromen-4-one
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
5-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
1-(3-propyl-1H-pyrazole-4-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
6-fluoro-4-(4-methyl-1,4-diazepane-1-carbonyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
2-(phenylsulfanyl)-N-[1-(pyridine-4-carbonyl)azepan-3-yl]acetamide
N-[3-(pyridin-2-yl)propyl]-3-sulfamoylbenzamide
4-[7-(furan-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]thiomorpholine
2-(dimethylamino)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2,3-dihydro-1H-indene-2-carboxamide
4-[(3,5-dimethoxyphenyl)methyl]-3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]piperazin-2-one
4-[4-ethyl-6-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]morpholine
5-chloro-N-(1-cyclopropanecarbonylpiperidin-3-yl)pyridine-2-carboxamide
1-(3-methoxyphenoxy)-3-{[4-(methylsulfanyl)butan-2-yl]amino}propan-2-ol
(2S,4S)-4-amino-N-ethyl-1-[1-(3-methylbutanoyl)piperidine-4-carbonyl]pyrrolidine-2-carboxamide
3-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,6-dichlorophenyl)urea
methyl 2-(benzylsulfamoyl)-6-[(4-hydroxyphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(4-acetylphenoxy)-N-(5-hydroxyadamantan-2-yl)acetamide
4-{5-methoxy-2-[(2-methoxyethyl)carbamoyl]phenoxy}-N,N-dimethylpiperidine-1-carboxamide