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4-(3-chloro-2-fluorobenzoyl)-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
ethyl 4-{1-[2-(methylsulfanyl)acetyl]piperidin-3-yl}piperazine-1-carboxylate
3-({[3-(1H-1,2,3-benzotriazol-1-yl)propyl]amino}methyl)pyrrolidin-3-ol
1-{2-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-oxoethyl}-1-methylurea
2-methoxy-5-{thieno[2,3-d]pyrimidin-4-yl}pyridine
N-[(4-ethylphenyl)methyl]-N-methyl-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-[(5-cyclopropyl-4-phenyl-1H-imidazol-1-yl)methyl]-3,5-dimethylpyridin-4-ol
1-cyclohexyl-4-[5-(phenoxymethyl)-1,2-oxazole-3-carbonyl]-1,4-diazepane
N-cyclopropyl-2,6-dimethoxy-N-{[4-(thiophen-3-ylmethoxy)phenyl]methyl}benzamide
2-[3-(methoxymethyl)phenyl]-2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}acetic acid
[(3R,4S)-1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
4-({4-methyl-5-[1-(2-methylpyrimidin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
4-[(3-methoxyphenyl)methyl]-N-[4-(methylsulfanyl)phenyl]-3-oxopiperazine-1-carboxamide
ethyl 4-[3-(4-methyl-4H-1,2,4-triazol-3-yl)propanoyl]piperazine-1-carboxylate
2-[(1-cyclobutanecarbonylpiperidin-4-yl)formamido]-2-(3-fluorophenyl)acetic acid
N-[(2-fluorophenyl)methyl]-4-(4-{[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]amino}piperidin-1-yl)benzamide
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-2-(methylamino)acetamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]acetamide
N-{2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}acetamide
N-[(4-{4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}phenyl)methyl]acetamide
3-benzoyl-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidine
4-(2-methoxyethyl)-3-[2-(4H-1,2,4-triazol-4-yl)ethyl]-4H-1,2,4-triazole
N-(1-benzothiophen-5-ylmethyl)-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-methyl-6-(2-phenylphenyl)pyridazine
(2E)-1-[3-(4-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxymethyl)piperidin-1-yl]-3-(thiophen-2-yl)prop-2-en-1-one
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-5,6-dimethylpyrimidin-4-amine
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)cyclohexanecarboxamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-5-(4-fluorophenyl)-1,2,4-triazin-3-amine
N-(2-{7-[(2,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methoxybenzamide
N-[2-(dimethylamino)ethyl]-N-methyl-1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}piperidin-3-amine
5-{3-[1-(cyclopropylmethyl)-1H-pyrazol-3-yl]phenyl}-N,N-dimethylfuran-2-carboxamide
1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-methyl-3-phenylpiperidine
8-[(2-aminopyridin-3-yl)methyl]-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-({[2-(dimethylamino)ethyl][(5-methylthiophen-2-yl)methyl]amino}methyl)-N-methylbenzene-1-sulfonamide
4-(2,3-dihydro-1H-inden-2-yl)-1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
3-{[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-5-methyl-1H-indole-2-carboxylic acid
2-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-1,2-oxazinane
1,5-dimethyl-4-{1-methyl-3-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrazole
5-chloro-N-cyclopropyl-3-methyl-N-({4-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-1H-indole-2-carboxamide
4-{[(2R)-2-hydroxypropyl]sulfamoyl}-N-[3-(methylsulfanyl)propyl]benzamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methylbenzamide
1-[1-({4-[methyl(phenyl)amino]phenyl}methyl)piperidin-3-yl]pyrrolidin-2-one
5-(4-fluorophenyl)-N-methyl-N-[3-(morpholin-4-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-(methylsulfanyl)-6-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl][(5-ethylpyridin-2-yl)methyl]methylamine
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[(2-fluorophenyl)methyl]-1,3-benzoxazole-6-carboxamide
1-[4-(furan-2-yl)butan-2-yl]-4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-3-azaspiro[5.5]undecan-9-amine
N-[(3S,4R)-1-[4-(4-chlorophenyl)butanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
[2-(dimethylamino)ethyl](methyl)(2-{[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]oxy}hex-5-en-1-yl)amine