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2-{[(5-ethylthiophen-3-yl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
4-[2-(propan-2-yl)pyrimidin-4-yl]-3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)urea
methyl (1R,3S,3aR,6aS)-3-(4,5-dimethylfuran-2-yl)-1-methyl-4,6-dioxo-5-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-1H-1,2,3-triazole-4-carboxamide
5-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
3-(azocan-1-yl)-N-(furan-2-ylmethyl)-N-(2-hydroxyethyl)propanamide
1-[3-({4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)phenyl]ethan-1-one
4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydroquinolin-2-one
dimethyl({4-[1-(5-methylpyridine-3-carbonyl)piperidin-2-yl]phenyl}methyl)amine
(1-{[1-(6-chloropyridazin-3-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
3-[(3R,4S)-3-amino-4-phenylpyrrolidine-1-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
methyl[(2-methyl-1,3-thiazol-4-yl)methyl]{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-1-(morpholin-4-yl)ethan-1-one
4-(1H-imidazol-1-ylmethyl)-1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-ol
3-(3-chloro-1,2-oxazol-5-yl)-1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]propan-1-one
(1R,3S,5S)-8-(2,3,5,6-tetramethylbenzoyl)-8-azabicyclo[3.2.1]octan-3-ol
5-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(2-methylpropanamido)benzamide
methyl 2-[(3,4-difluorophenyl)sulfamoyl]-6-(4-methylpentanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-2-(5-oxopyrrolidin-2-yl)acetamide
7-{4-[1-(morpholin-4-yl)ethyl]phenyl}-3,4-dihydro-2H-1-benzopyran-4-one
N-cyclopentyl-N-({4-[(2-fluorophenyl)methoxy]phenyl}methyl)-2H-1,3-benzodioxole-5-carboxamide
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[3-(1H-imidazol-1-yl)propyl]benzamide
1-[(4-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]piperidin-4-ol
N-{[3-methyl-7-(quinoxaline-6-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
4-(1-methyl-1H-pyrazole-5-carbonyl)-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
methyl[(4-phenyl-1,3-thiazol-2-yl)methyl][1-(pyrazin-2-yl)propan-2-yl]amine
2-[cyclopentyl(methyl)amino]-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}acetamide
(3R,4R)-1-(3-cyclopentylpropyl)-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
3-methyl-N-[2-(pyridin-4-yl)ethyl]-2-[(quinazolin-4-yl)amino]butanamide
2-(1H-pyrazol-1-yl)-1-{3-[4-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenoxymethyl]piperidin-1-yl}ethan-1-one
2-(2-hydroxyethyl)-8-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
(2S,4R)-4-(cycloheptylamino)-N-methyl-1-(propan-2-yl)pyrrolidine-2-carboxamide
2-methoxy-5-{[4-(1-methylpiperidin-4-yl)piperazin-1-yl]methyl}benzoic acid
N-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-methylpropyl]-4-(3-hydroxy-3-methylbutyl)benzamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-[(2-methoxyphenyl)methyl]-1-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide
2-(3-{[cycloheptyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)acetamide
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(phenylsulfanyl)acetamide
3-{4-[2-amino-6-methyl-5-(prop-2-en-1-yl)pyrimidin-4-yl]piperazin-1-yl}phenol
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
N-{[1-(carbamoylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}-2,4-dichlorobenzamide
(4aR,8aR)-2-methanesulfonyl-7-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-decahydro-2,7-naphthyridin-4a-ol
methyl 2-{[3-(2-methoxybenzoyl)piperidine-1-carbonyl]amino}benzoate
4-(4-benzyl-1H-pyrazol-5-yl)-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
(3S,4R)-4-(3-fluorophenyl)-1-(furan-3-ylmethyl)pyrrolidine-3-carboxylic acid
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(pyridin-3-ylmethyl)amine
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(1-methylpiperidin-4-yl)pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-ethylpyridin-2-yl)methyl]-N-methylacetamide
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2-methyl-4-(4-methylphenyl)piperazine