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1-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
1-[1-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)ethyl]-4-methylpiperazine
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-2,8-dimethylquinoline-4-carboxamide
3-benzyl-N-(oxan-4-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
2-methyl-2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}(thiophen-3-ylmethyl)amino)propan-1-ol
4-[(2-hydroxyethyl)sulfanyl]-N-methyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]benzamide
1-(cyclohexylmethyl)-N3,N3-dimethyl-4-oxo-N5-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-(1-ethylpiperidin-4-yl)-N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]acetamide
1-(2-chlorophenyl)-3-cyclopropyl-5-[(3-methyl-1H-pyrazol-1-yl)methyl]-1H-1,2,4-triazole
6-ethyl-4-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-2-methylquinoline
1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-[(4-ethyl-1,3-thiazol-2-yl)methyl]urea
7-(1,3-benzothiazol-2-yl)-4-(1,3-thiazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-N-[2-(1H-pyrazol-1-yl)ethyl]benzene-1-sulfonamide
3-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydroquinoxalin-2-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-methyl-4-[4-({2-methyl-2,8-diazaspiro[4.5]decan-8-yl}methyl)phenyl]butan-2-ol
1-(3-methoxypropyl)-3-[2-(phenylsulfanyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
(2S)-2-({[2-(benzyloxy)phenyl]carbamoyl}amino)-4-methylpentanamide
4-[1-(3-methylbutyl)-5-[2-(thiophen-2-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperazin-2-one
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-(morpholin-3-yl)acetamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
N-(4-fluorophenyl)-1-(4-methylpyridine-3-carbonyl)piperazine-2-carboxamide
N-({7-[(2,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
2-methyl-1-[(1-methyl-1H-imidazol-5-yl)methyl]-4-(2-methylphenyl)piperazine
1-[(1-methyl-1H-imidazol-2-yl)methyl]-8-(2-methylquinolin-4-yl)-1,8-diazaspiro[4.5]decane
2-{[4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-5-methoxyphenol
N-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylfuran-2-carboxamide
5-(2-chlorophenyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}furan-2-carboxamide
N-[(3R,4R)-3-hydroxy-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-4-yl]pyridine-3-carboxamide
N-(2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}phenyl)-5-methylfuran-2-carboxamide
(3R,5S)-N-{1-[(2-methylphenyl)methyl]cyclopropyl}-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}oxolane-3-carboxamide
N-(1H-1,3-benzodiazol-2-yl)-2-{[1-(1H-1,2,4-triazol-5-yl)ethyl]amino}acetamide
dimethyl[3-({5-[4-(morpholin-4-yl)phenyl]pyridin-2-yl}oxy)propyl]amine
(3S,4S)-1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-4-(propan-2-yloxy)pyrrolidin-3-ol
N-benzyl-2-(3-methyl-1,2-oxazol-5-yl)-N-[(4-methyl-1,3-thiazol-5-yl)methyl]acetamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-({[(3R,4R)-1-(5-fluoro-1-methyl-1H-indole-2-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
(2S,4R)-4-(3-methoxy-2-methylbenzamido)-N-methyl-1-(oxan-4-yl)pyrrolidine-2-carboxamide
4-benzyl-3-ethyl-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1,4-diazepan-5-one
2-(2H-1,3-benzodioxol-5-yl)-N-[1-(4-methylpyridin-2-yl)propyl]acetamide
N-({4-hydroxy-1-[2-(1H-indol-3-yl)acetyl]azepan-4-yl}methyl)methanesulfonamide
(4aR,8aR)-7-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
11-(6-hydroxy-2,6-dimethylheptyl)-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
N-[2-(dimethylamino)ethyl]-5-(4-phenylazepane-1-carbonyl)pyridin-2-amine
(2R,6R)-4-[2-methyl-2-(morpholin-4-ylmethyl)propyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(3S,4R)-3-(dimethylamino)-N-(2-phenylethyl)-4-(propan-2-yl)pyrrolidine-1-carboxamide
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-3-(piperidin-1-ylmethyl)piperidine