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(3aR,6aR)-2-acetyl-5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[(2-fluoro-5-methoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}({[4-(trifluoromethoxy)phenyl]methyl})amine
4,5-dimethyl-6-{4-[2-(pyrrolidin-1-yl)ethyl]piperazin-1-yl}pyrimidine
8-(2H-1,3-benzodioxol-5-ylmethyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
(1S,5R)-6-methyl-3-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[2-(3-phenylprop-2-ynoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-2-carboxamide
5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-4-methylpyrimidine
1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-N-(3,4-dimethylphenyl)piperidin-3-amine
3-(pyridin-3-ylmethoxy)-N-(5,6,7,8-tetrahydronaphthalen-1-yl)piperidine-1-carboxamide
N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
2-hydroxy-4-methyl-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pentanamide
(4aS,8aR)-6-(2-aminopyrimidin-4-yl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(oxan-4-ylmethyl)propanamide
2-amino-4-[3-(dimethylamino)pyrrolidin-1-yl]quinazoline-6-carboxylic acid
5-{2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-ethyl-5-methyl-1,2-oxazole-4-carboxamide
4-(4-{1-[(2-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}benzoyl)morpholine
N-{2-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
5-(3-{4-[(4-fluorophenyl)sulfanyl]piperidin-1-yl}-3-oxopropyl)-5-(thiophen-2-ylmethyl)pyrrolidin-2-one
N-(1-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}pyrrolidin-3-yl)acetamide
1-(but-2-yn-1-yl)-4-(1-phenyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridine
2-[4-(6-aminopyridine-3-carbonyl)piperazin-1-yl]-N-ethylacetamide
N,N-dimethyl-2-{[3-(1-methyl-1H-pyrazol-4-yl)propanamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
4-{2-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
4-(1H-1,3-benzodiazole-5-carbonyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
3-methyl-7-(4-methyl-1H-imidazole-5-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-(4-{4-[2-(3-hydroxypropyl)piperidine-1-carbonyl]phenoxy}piperidin-1-yl)-3-methoxypropan-1-one
(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-5-[3-(methylsulfanyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[2-(2-fluorophenoxy)ethyl]-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-3-(pyridin-3-yl)propanamide
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine
N-cyclopropyl-2-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
5-benzenesulfonamido-1-ethyl-N-(2-hydroxybutyl)-2-methyl-1H-1,3-benzodiazole-7-carboxamide
(2S,4R)-N,N-diethyl-1-(2-methylpropanoyl)-4-[2-(thiophen-2-yl)acetamido]pyrrolidine-2-carboxamide
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
(1R,3S,5S)-8-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
4-{5-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]pyrimidin-2-yl}morpholine
3-[methyl({[1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-5-yl]methyl})amino]-1λ6-thiolane-1,1-dione
2-{1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazol-2-yl}-1H-1,3-benzodiazole
4-benzyl-3-ethyl-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-1,4-diazepan-5-one
4-benzyl-1-(cyclopropylmethyl)-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2-(pyridin-2-ylsulfanyl)acetamide
N'-cyclopentyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}butanediamide
N-[3-(1H-indol-1-yl)propyl]-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
6-methoxy-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-methoxy-2-phenyl-1-{4-[5-phenyl-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one