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3-{1-[(4-phenylphenyl)methyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-(2-hydroxyethyl)-8-methoxy-N-[(3-methylthiophen-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-(3-methoxypropyl)-N-(quinolin-5-yl)piperazine-1-carboxamide
N-(4-fluoro-2-methylphenyl)-3-[1-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)piperidin-3-yl]propanamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-{4-[(5-ethylpyridin-2-yl)methyl]morpholin-3-yl}-N-methylacetamide
1-(cyclobutylmethyl)-3-hydroxy-3-(morpholin-4-ylmethyl)piperidin-2-one
1-{[(4-chloro-2-methoxy-5-methylphenyl)carbamoyl]amino}cycloheptane-1-carboxamide
3-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
3-[(dimethylamino)methyl]-1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]piperidin-3-ol
2-{4-[(3,5-dimethoxyphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
methyl (2S,4R)-4-cyclohexaneamido-1-[(2-fluorophenyl)methyl]pyrrolidine-2-carboxylate
2-(piperidin-1-yl)-5-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)pyrimidine
2-(dimethylamino)-2-(2-fluorophenyl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
[(1-cyclopentylpiperidin-4-yl)methyl][(1-ethyl-1H-pyrazol-4-yl)methyl](pyridin-3-ylmethyl)amine
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)(methyl)[(3-methylpyridin-4-yl)methyl]amine
7-methyl-4-(morpholine-4-carbonyl)-2-[2-(propan-2-yl)pyrimidin-5-yl]quinoline
2-{[(6,8-dimethyl-2-oxo-2H-chromen-4-yl)methyl]amino}-N,N-dimethylethane-1-sulfonamide
2-amino-4-(2-chloro-4-hydroxyphenyl)-6-(trimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
(4aR,7aS)-1-cyclopropanecarbonyl-4-[(4-hydroxy-3,5-dimethylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3aR,7aS)-5-methyl-2-[4-(1H-pyrazol-3-yl)benzoyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
4-(piperidin-1-yl)-1-[4-(pyridin-3-yl)pyrimidin-2-yl]piperidine-4-carboxamide
2-[5-(2,6-difluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
1-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}-4-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazine
3-{2-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydro-1,2,3-benzotriazin-4-one
1-(pyrazin-2-yl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,4-diazepan-6-ol
3-(3,4-dimethylphenyl)-4-{1H-imidazo[4,5-b]pyridin-2-yl}-1H-pyrazole
1-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazole
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(benzyloxy)ethan-1-one
1-cycloheptyl-1-methyl-3-(1,3,4-thiadiazol-2-yl)urea
1-(2,3-difluoro-6-methoxybenzoyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
1-(2-methoxyphenyl)-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazin-2-one
{[(3S,4R)-1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
N-benzyl-3-({1-[1-(pyridin-3-yl)propan-2-yl]piperidin-4-yl}oxy)benzamide
N-(3-hydroxy-3-phenylpropyl)-N-methylpyrazolo[1,5-a]pyridine-7-carboxamide
N-(oxan-3-yl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
5-(oxolan-2-yl)-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}thiophene-2-carboxamide
1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
1-({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)-2-(1,3-thiazol-2-yl)piperidine
1-[4-(propan-2-yl)-1,2,3-thiadiazole-5-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxylic acid
[(2,4-dimethoxyphenyl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
1-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
N-[2-(pyrazin-2-yl)ethyl]-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-ethyl-1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
dimethyl({4-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1,3-thiazol-2-yl}methyl)amine
(1-{7-[(cyclopentylamino)methyl]-2H-[1,3]dioxolo[4,5-g]quinolin-6-yl}piperidin-3-yl)methanol
N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetamide
1-[2-(2,4-dimethylphenoxy)ethyl]-4-ethyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N4-(1-tert-butyl-4-phenyl-1H-pyrazol-5-yl)morpholine-2,4-dicarboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine