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2-(cyclopropylmethyl)-8-(2-methyl-5-propylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
3-(3-methoxyphenoxy)-1-[4-(5-methylfuran-2-yl)benzoyl]azetidine
5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-1-[3-(morpholin-4-yl)propyl]piperidin-2-one
N-[(3R,4R)-3-hydroxy-1-(3,3,3-trifluoropropyl)piperidin-4-yl]pyridine-2-carboxamide
[1-(2-{[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]amino}ethyl)piperidin-2-yl]methanol
3-[3,5-dimethyl-1-(1-oxo-2,3,4,9-tetrahydro-1H-carbazol-6-yl)-1H-pyrazol-4-yl]propanoic acid
3-(2H-1,3-benzodioxol-5-yl)-N-[(6-methylpyridin-2-yl)methyl]-3-phenylpropanamide
3-(5-fluoro-2-methoxybenzoyl)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidine
methyl 1-{3-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1,2-oxazole-5-carbonyl}piperidine-4-carboxylate
5-ethyl-3-(pyridin-2-ylmethyl)-5-{1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}imidazolidine-2,4-dione
2-(propan-2-yloxy)-1-{spiro[azepane-4,2'-chromene]-1-yl}ethan-1-one
methyl 7-oxo-3-[2-(1,3-thiazol-4-yl)acetyl]-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(4aS,8aR)-1-butyl-6-(2-oxo-2,3-dihydro-1H-imidazole-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
4-{[9-(2-methoxyethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl]methyl}-N-methylbenzamide
1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
2-({3-[4-(5-cyanopyridin-2-yl)piperazine-1-carbonyl]phenyl}amino)acetic acid
3-{[ethyl(methyl)amino]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-{1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]piperidin-4-yl}piperidin-4-ol
2-[(2-hydroxyethyl)({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]ethan-1-ol
1-methyl-10-oxo-9-(prop-2-en-1-yl)-N-propyl-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
5-{[3-(3-methoxypropyl)piperidin-1-yl]methyl}-1H-indole
2-{5-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-1-yl}acetic acid
3-[1-(cyclopent-3-ene-1-carbonyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
N-[3-(1H-pyrazol-1-yl)phenyl]imidazo[1,2-a]pyrimidine-2-carboxamide
5-(2-methylpropyl)-5-[1-(quinoxalin-5-ylmethyl)piperidin-4-yl]-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
3-({[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)-N,N-dimethylthiolan-3-amine
N-[(4-methylphenyl)methyl]-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
2-{[(2-hydroxy-4-methylphenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-[2-(morpholine-4-carbonyl)piperazin-1-yl]-3-phenoxypropan-1-one
methyl (2R,4S)-4-hydroxy-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine-2-carboxylate
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[(1R)-1-(4-methoxyphenyl)ethyl]amino}piperidin-1-yl)benzamide
N-methyl-5-{[2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamido]methyl}-1,2,4-oxadiazole-3-carboxamide
5-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
N-(1-{7-[(5-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
N-(1-methyl-1H-pyrazol-4-yl)-2-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}acetamide
N3-benzyl-1-cyclopropyl-N5-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-ethyl-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
4-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-1-phenylpiperazin-2-one
2-{4-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}pyrimidine
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-{[1-(morpholin-4-yl)cyclohexyl]methyl}pyrrolidin-2-one
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-oxo-1,4-dihydroquinoline-2-carboxamide
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
7-(5-chloropyridin-2-yl)-9-methoxy-4-[4-(trifluoromethyl)benzenesulfonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[(4-fluorophenyl)methyl]-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1,2-oxazole-5-carboxamide
N-{1-[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N,3-dimethylbutanamide
1-[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-propylpentan-1-one
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-4-(pyridin-2-yl)pyrimidin-2-amine
2-(adamantan-1-yl)-4-hydroxy-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]pyrimidine-5-carboxamide
1-(3-methylfuran-2-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
3-[(3S,4R)-3-cyclopropyl-4-(2-ethoxybenzamido)pyrrolidin-1-yl]propanoic acid