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2-{1-[(1,3-dimethylpyrrolidin-3-yl)methyl]-1H-imidazol-2-yl}-1-(4-methoxyphenyl)-1H-imidazole
N-methyl-1-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N,N-diethyl-1-[1-(2-methylpropyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
2-[1-(2H-1,3-benzodioxol-5-yl)-5-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-yl)-1H-1,2,4-triazol-3-yl]acetamide
2-[1-(pyrimidin-2-yl)azetidin-3-yl]-1H-1,3-benzodiazole
(2R)-1-{[2-(3-chlorophenyl)-7-fluoroquinolin-3-yl]methyl}pyrrolidine-2-carboxamide
4-(thiophen-2-ylsulfanyl)-6-[2-(trifluoromethyl)morpholin-4-yl]pyrimidin-2-amine
1-{[1-(3-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazol-5-amine
3-[3-(azepane-1-carbonyl)phenyl]-1-[1-(pyridin-3-yl)propyl]urea
2-(4-methoxyphenoxymethyl)-N-[(1r,4r)-4-hydroxycyclohexyl]-1,3-oxazole-4-carboxamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-(3-methylthiophene-2-carbonyl)pyrrolidin-3-yl]methanol
2-(3-fluorophenoxymethyl)-N-(2-hydroxy-3-methoxypropyl)-1,3-oxazole-4-carboxamide
(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-7-[(thiophen-3-ylmethyl)amino]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(3S,4R)-1-(2-methanesulfonamidoacetyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
(2S,4S)-N-cycloheptyl-1-[(2E)-3-phenylprop-2-en-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-[(3-phenyl-1H-pyrazol-4-yl)methyl]-decahydro-2,7-naphthyridine-2-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-N-(furan-3-ylmethyl)piperidin-3-amine
4-(2,6-dimethylpyridin-3-yl)-2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}pyrimidine
2-[3-(pyridin-2-yl)azetidin-1-yl]-4-(trifluoromethyl)pyridine
methyl 9-(cyclopentyloxy)-3-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-5-methylpyrazine
1-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazole
1-[(4-chlorophenyl)methyl]-N-methyl-N-(oxan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-{4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}ethan-1-one
2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]acetamide
6-methyl-2-oxo-N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)-4-(thiophen-2-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-5-methylpyridine
(4aS,7aR)-1-(2-hydroxybenzoyl)-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-4-(pyrrolidin-1-ylmethyl)benzamide
3-[({2-[2-(trifluoromethoxy)phenyl]ethyl}amino)methyl]piperidin-3-ol
2-(2,4-dichlorophenoxy)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)acetamide
N,2,2-trimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1-(thiophen-2-yl)cyclopropane-1-carboxamide
N-(2-methylpropyl)-1-[1-(quinolin-4-ylmethyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
6-cyclopentyl-1-methyl-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4,6-dimethyl-1-{2-oxo-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethyl}-1,2-dihydropyrimidin-2-one
1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-[3-(methylsulfanyl)propyl]piperidine-4-carboxamide
5-(oxolan-2-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}thiophene-2-carboxamide
N-[4-(3-methylphenyl)phenyl]-1-[(3-methylquinoxalin-2-yl)methyl]piperidine-4-carboxamide
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]pyrrolidin-3-yl]urea
N-{[7-(2,3-dihydro-1-benzofuran-5-ylmethyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(phenylsulfanyl)acetamide
2-butyl-N-(4-methanesulfonylphenyl)-4-methyl-3-oxopiperazine-1-carboxamide
3-phenyl-1-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidin-4-yl)propan-1-ol
2-(3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzoyl)-1,2,3,4-tetrahydroisoquinoline
[(3S,5R)-1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
N-methyl-N-[2-phenyl-1-(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)ethyl]thiophene-3-carboxamide
4-[2-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyridine-4-carbonyl]morpholine
2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-[2-(pyrrolidin-1-yl)ethyl]-1H-imidazole
N-(cyclopropylmethyl)-2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
1-(4-{4-phenyl-1-[2-(pyridin-2-yl)ethyl]-1H-imidazol-5-yl}phenyl)ethan-1-one