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4-{4-[(2-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-1λ6-thiane-1,1-dione
2-(dimethylamino)-7-[5-(oxolan-2-yl)thiophene-2-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)imidazolidine-2,4-dione
7-(2-oxoimidazolidin-1-yl)-4-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1,2,3,4-tetrahydroquinolin-2-one
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-N-[2-methoxy-2-(thiophen-2-yl)ethyl]propanamide
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]-4-methyl-1,3-thiazole-5-carboxamide
9-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(3-methylbutyl)-8-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
(4S)-1-[(2,3-dimethoxyphenyl)methyl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
2-(3-methoxypropyl)-1-[2-(4-methylbenzoyl)benzoyl]piperidine
2-[1-(propan-2-yl)piperidin-4-yl]-N-[1-(pyrazin-2-yl)propan-2-yl]acetamide
N-[(2R,3R)-1'-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
5-(4-oxo-4H-chromene-2-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
3-[4-(3-methylphenyl)piperazin-1-yl]-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]propanamide
N-[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]-4-(4-chlorophenoxy)piperidine-4-carboxamide
N-propyl-N-(pyridin-3-ylmethyl)-1,3-benzothiazole-6-carboxamide
2-(isoquinolin-5-yl)-5-methylpyrimidin-4-amine
N-[(4-ethylphenyl)methyl]-2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-6-(1-methylpiperidin-3-yl)pyrimidin-4-amine
N-(propan-2-yl)-1-(2-{4-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperazin-1-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-(diethylamino)-3-[5-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
4-(3-methylbutyl)-3-{2-oxo-2-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethyl}piperazin-2-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(propan-2-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,3-benzoxazole-5-carboxamide
N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-1-(pyridin-2-ylmethyl)piperidin-4-amine
({3-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-1,2-oxazol-5-yl}methyl)(methyl)(2-phenylethyl)amine
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(1R,5S)-6-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}-6-azabicyclo[3.2.1]octane
2-methoxy-6-{[2-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenol
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylacetamide
5-{2-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(1H-imidazol-1-yl)-1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]butan-1-one
4-[4-(pyridin-3-yl)piperazin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
N-methyl-N-[(1R)-1-(naphthalen-1-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
9-(2-fluorobenzoyl)-1-methyl-4-[(2E)-2-methylpent-2-en-1-yl]-1,4,9-triazaspiro[5.5]undecane
methyl 3-(4-methoxybenzamido)-1-methyl-5-[(2-methylpropyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(3aR,7aS)-2-(5-methoxyfuran-2-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
(1S,5R)-6-(2-methoxyethyl)-N-methyl-7-oxo-N-phenyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-({3-[2-(4-fluorophenoxy)ethyl]phenyl}methyl)acetamide
methyl[(3-{2-[4-(2,3,4,9-tetrahydro-1H-carbazole-6-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](1,3-thiazol-4-ylmethyl)amine
[1-(1H-1,3-benzodiazol-2-ylmethyl)-3-(2-phenylethyl)piperidin-3-yl]methanol
(1S,5R)-6-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
methyl 5-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-{4-[methyl({[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl})amino]piperidin-1-yl}ethan-1-one
2-[5-(1,5-dimethyl-1H-pyrrole-2-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(4-fluorophenyl)piperazine-2-carboxamide
1,3-dimethyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine