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N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
(3S,5R)-N3-cyclopropyl-N5-(4-fluorophenyl)-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
3-(1-cycloheptylpiperidin-3-yl)-N-(2-fluorophenyl)propanamide
1-[(4-fluorophenyl)methyl]-4-(9H-purin-6-yl)piperazin-2-one
4-chloro-3-methyl-N-(prop-2-en-1-yl)-N-(propan-2-yl)benzamide
(3aS,6aS)-2-cyclobutanecarbonyl-5-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 4-(4-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
(1R,5R)-3-(5-fluoro-1-methyl-1H-indole-2-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
1-{1-[(2S,4S)-1-[(2-chlorophenyl)methyl]-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carbonyl]piperidin-4-yl}-4-ethylpiperazine
2-cyclobutaneamido-7-oxo-N,N-bis(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
methyl 3-[(2E)-3-phenylprop-2-enamido]-5-[(pyridin-2-ylformamido)methyl]benzoate
[(3S,5R)-1-[(3,4-difluorophenyl)methyl]-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
N,N-bis(2-hydroxyethyl)-N'-(4-methylphenyl)propanediamide
methyl 4-[(4-{2-[(2,4-dimethoxyphenyl)carbamoyl]ethyl}piperidin-1-yl)methyl]benzoate
3-{1-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinane-4-carbonyl]piperidin-4-yl}-N-phenylpropanamide
2-methoxy-N,N-bis(propan-2-yl)-6-(pyrazin-2-yl)benzamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(5-methylfuran-2-yl)methyl]pyrrolidin-3-yl]-5-hydroxypyrazine-2-carboxamide
1-(2-methoxyphenyl)-4-[2-(1H-pyrazol-1-yl)butanoyl]piperazin-2-one
3-[5-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}urea
2-(2-methoxyethoxy)-1-{4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl}ethan-1-one
3-{[3-(hydroxymethyl)-4-methylpiperazin-1-yl]methyl}-7-methyl-1,2-dihydroquinolin-2-one
1-cyclopentyl-4-(1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)piperazine
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(3-methylphenyl)acetamide
4-ethyl-6-{3-[(2-methylphenyl)methoxy]azetidin-1-yl}pyrimidine
1-ethyl-3-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-5-methyl-1H-pyrazole
2-[methyl({4-methyl-5-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
1-(2,3-dihydro-1H-inden-2-yl)-4-[(6-methoxypyridin-3-yl)methyl]-1,4-diazepane
methyl 9-[(1-methylpiperidin-3-yl)methoxy]-7-oxo-3-(quinolin-5-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[(diethylamino)methyl]-N,5-diethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]furan-2-carboxamide
2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
(1S,5R)-6-(2-methoxyethyl)-3-{[4-(propan-2-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
7-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
methyl 4-{[6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}butanoate
4-(1H-pyrazole-4-carbonyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
N-(pyridin-2-ylmethyl)-1-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-chloro-N,N-dimethyl-4-[({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}carbamoyl)amino]benzamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,2-dimethyl-1-benzofuran-7-carboxamide
2-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-6-methoxyphenol
2-(1-ethylpiperidin-4-yl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
8-[3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
5-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
2-{4-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-ylmethyl]phenyl}ethan-1-amine
3-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3,4-dimethylphenyl)urea
N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)-2H-1,3-benzodioxole-5-carboxamide
1,2-dimethyl-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazine
3-(4-chlorophenyl)-1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]propan-1-one
2-{[2-amino-7-(furan-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl](methyl)amino}-N-methylacetamide
5-chloro-3-[(1R,5S,8R)-8-methoxy-3-azabicyclo[3.2.1]octane-3-carbonyl]-1,2-dihydropyridin-2-one