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4-{4-phenyl-1-[4-(pyrrolidin-1-yl)butyl]-1H-imidazol-5-yl}pyridine
3-{[1-(2-methoxybutanoyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-6-methyl-1-(2-methylphenyl)piperazin-2-one
N,N-dimethyl-6-(3,4,5-trimethoxyphenyl)pyridine-2-carboxamide
(3S,9aR)-8-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-1H-pyrazole-3-carboxamide
2-(thiophen-2-yl)-N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}acetamide
(3R)-1-[4-(4-chlorophenoxy)piperidine-4-carbonyl]piperidin-3-ol
3-({1-[3-(2-oxopiperidin-1-yl)propanoyl]pyrrolidin-3-yl}methyl)benzoic acid
5-(4-chloro-2-methoxyphenoxymethyl)-N-(2-phenylpropyl)-1,2-oxazole-3-carboxamide
3-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]methyl}benzoic acid
methyl 2-[(2-methylphenyl)sulfamoyl]-6-(pent-4-enoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-benzyl-5-[(3-ethoxy-4-methoxyphenyl)methyl]-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{4-[(tert-butylamino)methyl]-2-methoxyphenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
3-(2-chlorophenyl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-phenylpropanamide
1-[2-({[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
({2-[(2-chloroprop-2-en-1-yl)oxy]-6,7-dimethoxyquinolin-3-yl}methyl)[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
1-cyclobutanecarbonyl-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1,4-diazepane
9-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-ethyl-9-(4-fluoro-2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S,4R)-1-{[4-(benzyloxy)phenyl]methyl}-N-(2-phenylethyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[1-(4-methylphenyl)propyl]benzamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]pyrrolidin-3-yl]methanol
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-({4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
1-[(2-chlorophenyl)methyl]-N-[1-(4-methoxyphenyl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-{4-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
5-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazole
ethyl 4-[(4-methoxyphenyl)methyl]-1-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}piperidine-4-carboxylate
2-[(4-methyl-1,3-thiazol-5-yl)methyl]-2-azaspiro[4.4]nonan-3-one
(3S,4R)-1-(2,4-dichlorobenzenesulfonyl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-[2-(2-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[(2-fluorophenyl)methyl]-1-methyl-5-{[(3-methyloxetan-3-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[2-(4-fluorophenyl)ethyl]-N-({2-[3-(hydroxymethyl)piperidin-1-yl]-7-methoxyquinolin-3-yl}methyl)-2-methylpropanamide
5-[1-(2,5-difluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1-ethyl-3-methyl-1H-pyrazole
N-methyl-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]acetamide
N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-(4-chloro-3-methylphenyl)-1-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]urea
1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-methyl-1,4-diazepan-5-one
N-methyl-3-[(2-methylprop-2-en-1-yl)oxy]-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
N-({5-[(4-fluoro-3-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
2-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
2-({4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}methyl)quinolin-4-ol
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}acetamide
2-(2-methyl-1,3-thiazol-4-yl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]acetamide
methyl 2-[(cyclohexylmethyl)sulfamoyl]-6-(2,2-dimethylpropanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(4-chlorobenzoyl)-4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
(5S,9aS,9bS)-2-(2-methoxyphenyl)-5-[4-(propan-2-yl)-1,3-thiazol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one