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2-(2H-1,3-benzodioxol-5-yl)-N-{imidazo[1,2-a]pyrazin-3-ylmethyl}acetamide
(2S)-1-(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)pyrrolidine-2-carboxamide
4-methoxy-6-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
1-methyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H-imidazole-4-sulfonamide
3-[methyl(pyrazin-2-ylmethyl)sulfamoyl]-N-phenylbenzamide
N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)acetamide
[(3S,7S)-5-cyclobutanecarbonyl-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-trien-3-yl]methanol
methyl({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl){[4-(trifluoromethoxy)phenyl]methyl}amine
3-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-N-cyclohexyl-N-methylpyridin-2-amine
methyl 3-(2-methylbutanamido)-1-(oxolan-2-ylmethyl)-5-[(thiolan-3-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(2-ethylphenyl)-2-(2-methanesulfonylacetamido)benzamide
methyl 1-(2-methoxyethyl)-5-[(pentan-3-yl)amino]-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(2S)-1-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}pyrrolidine-2-carboxamide
(1H-indol-4-ylmethyl)({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
N-methyl-N-[2-(4-methylphenoxy)ethyl]-6-(thian-4-yl)-6-azaspiro[2.5]octane-1-carboxamide
N-[2-(2-methoxyphenyl)ethyl]-6-{[4-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
7-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl 3-(2H-1,3-benzodioxol-5-ylmethyl)-9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{[2-(4-chlorophenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}piperidin-4-ol
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-4-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-1,3-oxazole
N,N-bis(1,3-oxazol-4-ylmethyl)-4-(1H-pyrazol-3-yl)benzamide
1-(cyclopropylmethyl)-5-[(5-acetamidothiophen-2-yl)methyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(4-aminoazepane-1-carbonyl)-1-methyl-1,2-dihydropyridin-2-one
(1S,5R)-3-{[4-(methylsulfanyl)phenyl]methyl}-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(4-{[1-benzyl-2,4-dioxo-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}phenyl)acetamide
(4aS,8aR)-6-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
6-{4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}pyridine-2-carbonitrile
3-fluoro-2-methoxy-N-[1-(thiophen-2-yl)propyl]benzamide
1-[(2,6-dimethylphenyl)methyl]-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(1R,3S,5S)-8-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-{6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridazin-3-yl}thiomorpholine
N,N-diethyl-1-(2-methylpyrimidine-5-carbonyl)pyrrolidin-3-amine
(2S)-N-[3-chloro-4-(1H-imidazol-1-yl)phenyl]-2-(methoxymethyl)pyrrolidine-1-carboxamide
N-(2-methylpropyl)-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
7-[(2,3-difluorophenyl)methyl]-2-(2,5-dimethylfuran-3-carbonyl)-2,7-diazaspiro[4.5]decane
N-[(4-methoxy-2,3-dimethylphenyl)methyl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
(2R,6S)-4-[1-(6-methoxypyrimidin-4-yl)piperidin-4-yl]-2,6-dimethylmorpholine
N-{1-[4-(3-phenylpiperidine-1-carbonyl)phenyl]-1H-pyrazol-4-yl}pyridine-3-carboxamide
N-{2-[7-(1-benzothiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-(4-fluorophenyl)acetamide
6-chloro-2-(1-{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
N-{1-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-1H-pyrazol-4-yl}-2-(phenylsulfanyl)acetamide
2-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]acetic acid
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
(dicyclopropylmethyl)(methyl){[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}amine
2-{2-[(butan-2-yl)amino]ethyl}-6-phenyl-2,3-dihydropyridazin-3-one
3-{[(2-methoxyethyl)(1,3-thiazol-2-ylmethyl)amino]methyl}pyrrolidin-3-ol
N-{5-chloro-2-[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidine-1-carbonyl]phenyl}propanamide
1-(2,3-dihydro-1H-inden-2-yl)-5-[(3,4,5-trimethoxyphenyl)methyl]-1H-1,2,4-triazole
[(1-cyclohexylpiperidin-3-yl)methyl][(3-methyl-1,2-oxazol-5-yl)methyl](pyridin-3-ylmethyl)amine