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5-(diethylamino)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(3-cyanopiperidine-1-carbonyl)-N-(2-fluoroethyl)benzene-1-sulfonamide
1-cyclopentyl-3-(2-methoxyphenyl)-3-(2-oxo-2-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl}ethyl)pyrrolidine-2,5-dione
5-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-[(2-chlorophenyl)methyl]-3-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]propanamide
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(thiophen-3-ylmethyl)piperidine
N-cyclohexyl-3-[(1,3-thiazol-2-ylmethyl)sulfamoyl]benzamide
N-{[1-(1-benzofuran-2-carbonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
2-(furan-2-yl)-2-oxo-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
N-{2-[7-(3-phenylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}cyclohexanecarboxamide
methyl 3-(3-fluorobenzoyl)-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[(5-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]-3,3-dimethylurea
3-[3-(dimethylamino)propyl]-5-[(4-fluorophenyl)methyl]-5-[1-(2-methylbutyl)piperidin-4-yl]imidazolidine-2,4-dione
6-methyl-3-[4-oxo-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,2-dihydropyridin-2-one
1-phenyl-N-{2-[(2E)-3-(pyridin-3-yl)prop-2-enoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}cyclopropane-1-carboxamide
(3aS,6aS)-2-methyl-5-[(1-propyl-1H-pyrazol-5-yl)sulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-5-[(2-oxo-5,5-diphenylpiperidin-1-yl)methyl]furan-2-carboxamide
4-[3-(1H-indazol-1-yl)propyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-3,3-diphenylpiperidine
2-chloro-5-(piperidin-1-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}benzamide
2-{4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-2-oxopiperazin-1-yl}benzonitrile
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
[(3R,4R)-1-[(5-ethylfuran-2-yl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
7-(dimethyl-1,3-thiazole-5-carbonyl)-2-oxa-7-azaspiro[4.5]decane
5-(4-methylpyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline
4-[6-(1-benzofuran-2-yl)pyridine-3-carbonyl]morpholine
2-(2-{4-[(3,5-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-5,6-dimethyl-2,3-dihydropyridazin-3-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]acetamide
4-[(2-methyl-1H-imidazol-4-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-cyclohexyl-N-(2-hydroxy-2-phenylethyl)-2-(propan-2-yl)pyrimidine-5-carboxamide
N-cyclopropyl-2-ethyl-N-(1H-indol-5-ylmethyl)-4-methyl-1,3-oxazole-5-carboxamide
2-(6-oxo-1,6-dihydropyrimidin-5-yl)-N-[3-(pyridin-2-yl)propyl]acetamide
4-{[7-benzyl-3-(oxan-4-yl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-5-yl]methyl}-1H-imidazole
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(4-phenylpiperidin-1-yl)acetamide
N-methyl-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
3-methoxy-1-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]piperidine
5-(adamantane-1-carbonyl)-3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-[2-methyl-5-(trifluoromethyl)benzoyl]piperidin-4-ol
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}oxan-4-amine
6,6-dimethyl-5-oxo-N-[3-(phenylsulfanyl)propyl]thiomorpholine-3-carboxamide
ethyl 4-benzyl-1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidine-4-carboxylate
(2S,4S)-N-(1-benzothiophen-2-ylmethyl)-1-[(2-chloro-6-fluorophenyl)methyl]-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-N-methylpyrrolidine-2-carboxamide
1-propyl-5-[4-(pyridin-4-yl)-1,4-diazepan-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
4-{1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-methylpropan-2-yl}morpholine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(2-methylphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(1-{5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidin-2-yl)pyridine
9-[3-(2-fluorophenyl)-3-phenylpropanoyl]-2,9-diazaspiro[5.5]undecan-3-one
(4aS,7aR)-1-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[4-(1-benzyl-1H-pyrazol-4-yl)-1H-pyrazol-1-yl]-N-methylacetamide
6-ethyl-3-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-3,4-dihydroquinazolin-4-one