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N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
6-[2-(benzenesulfonyl)ethyl]-5,6-dihydro-1,6-naphthyridin-5-one
N-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}-1,2,3,4-tetrahydronaphthalen-1-amine
2-(4-phenylpiperidin-1-yl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]acetamide
5-(2,6-dimethylbenzoyl)-1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
N-[1-benzyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
N-(2-ethylphenyl)-3-[(pyrrolidin-3-yl)sulfamoyl]benzamide
2-(4-cyclopentyl-1,4-diazepane-1-carbonyl)-5-fluoro-1,3-dimethyl-1H-indole
9-hydroxy-2-{[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
8-{2-[2-(butan-2-yl)phenoxy]acetyl}-2,8-diazaspiro[4.5]decan-3-one
methyl 6-[1-(3-methoxyphenyl)propan-2-yl]-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(2-methoxy-4-{[methyl(oxan-4-ylmethyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
1-{3-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]piperidin-1-yl}ethan-1-one
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-methoxyethan-1-one
ethyl 2-[2-({1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-methyl-1H-pyrazol-4-yl}formamido)ethyl]-1,3-thiazole-4-carboxylate
4-benzyl-3-ethyl-1-[2-(piperidin-1-yl)acetyl]-1,4-diazepan-5-one
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-[2-(4-methoxybenzoyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
4-(2H-1,3-benzodioxol-5-ylmethyl)-2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
8-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N'-(3-ethylphenyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}butanediamide
N,N-dimethyl-1-[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]azepan-4-amine
5-[3-(1H-imidazol-1-yl)propyl]-3-(oxolan-3-yl)-1-propyl-1H-1,2,4-triazole
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-(piperidin-3-yl)benzamide
4-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,4-oxazepane
N-benzyl-2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-(oxolan-2-ylmethyl)acetamide
1-{3-methyl-5-[2-(4-methylphenyl)ethyl]-1H-1,2,4-triazol-1-yl}butan-2-ol
N-[2-(4-methylpiperidin-1-yl)ethyl]-N-(propan-2-yl)pyridine-3-carboxamide
N2-benzyl-6-(2,4-dichlorophenyl)-1,3,5-triazine-2,4-diamine
N-[1-(cyclohexylmethyl)-1H-pyrazol-5-yl]-4-(pyrazin-2-yl)piperazine-1-carboxamide
1-(4-{3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-one
N-(2-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]formamido}ethyl)pyridine-3-carboxamide
N-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-5-(hydroxymethyl)furan-2-carboxamide
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4,4,4-trifluorobutanamide
(3S,4R)-4-phenyl-1-[4-(1H-pyrazol-4-yl)butanoyl]pyrrolidine-3-carboxylic acid
2-[1-(1-methylpiperidin-4-yl)piperazin-2-yl]ethan-1-ol
1-butyl-3-methyl-4-(1-methyl-1H-indol-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
2-[4-(4-ethoxypyrimidin-2-yl)piperazin-1-yl]-N-(propan-2-yl)acetamide
N-(dicyclopropylmethyl)-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-methylpropanamide
5-methoxy-1-methyl-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-1H-indole-2-carboxamide
1-(furan-2-ylmethyl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidine-3-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-2-(furan-2-yl)-2-oxo-N-(oxolan-2-ylmethyl)acetamide
3-{[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]piperidine-1-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}propanamide
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
4-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,2,2-trimethylpiperazine
3-(4-fluorophenyl)-N-{3-[methyl(phenyl)amino]propyl}-1H-pyrazole-5-carboxamide
2-ethyl-9-(quinolin-6-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[2-methoxy-5-(3-methylpiperidine-1-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one