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1-{1-[4-(pyridin-3-yl)pyrimidin-2-yl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-methoxy-N-({8-[(4-methoxynaphthalen-1-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]acetamide
2,3-dimethyl-7-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-[4-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
1-{3-[2-(pyridin-2-yl)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
methyl (2S,4R)-4-(2-fluorobenzamido)-1-[(3-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxylate
8-[(4-ethynylphenyl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
3-[(3R,4S)-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(3S,9aR)-3-(1H-indol-3-ylmethyl)-8-[4-(trifluoromethyl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
8-(2,2-dimethylpropyl)-3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-6-(piperidin-4-yl)pyrimidin-4-amine
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-hydroxybutanamide
5-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2-methoxyphenol
3-(5-fluoro-2-methoxybenzoyl)-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidine
N-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-4-phenylbenzamide
(1R,4S)-N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-4-carboxamide
N-(1-{7-[(3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
4-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]-2-(pyridin-4-yl)quinoline
ethyl 3-[(3-chlorophenyl)methyl]piperidine-3-carboxylate
5-(1H-indol-1-ylmethyl)-N-[1-(pyrimidin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
1-[(4-methylphenyl)methyl]-4-(3-propyl-1,2,4-oxadiazol-5-yl)pyrrolidin-2-one
4-{4-[(1E)-pent-1-en-1-yl]phenyl}piperidin-4-ol
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-{4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}-1-methylpiperazin-2-one
methyl 4-(3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}propanamido)butanoate
N-({7-[(3-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
N-(1-methanesulfonylpiperidin-4-yl)-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
2-{4-[(2-methyl-1,3-thiazol-5-yl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
2-(4-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-1-(2,2-dimethylpropyl)piperazin-2-yl)ethan-1-ol
N-(3-methyl-1-{7-[(2,4,6-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)furan-2-carboxamide
N-(3-methoxy-3-methylbutyl)-6-(propan-2-yl)pyrimidin-4-amine
1-{5-[3-(methoxymethyl)phenyl]-1H-1,2,4-triazol-1-yl}butan-2-ol
4-(1H-1,3-benzodiazol-1-yl)-1-[(5-methylfuran-2-yl)methyl]piperidine-4-carboxylic acid
N-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-3-(3-hydroxy-3-methylbutyl)benzamide
9-[(3-chloro-4-methoxyphenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 2-{4-[({[1-(hydroxymethyl)cyclopentyl]methyl}carbamoyl)amino]phenoxy}acetate
1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(3-methoxypropyl)piperidine
(1S,5R)-3-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3R,4S)-4-(3-methoxyphenyl)-1-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-amine
(3aR,5S,6S,7aS)-2-(7-chloro-4-hydroxyquinoline-3-carbonyl)-octahydro-1H-isoindole-5,6-diol
{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}(ethyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
1-[(2-fluorophenyl)methyl]-5-[4-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]piperidin-2-one
(1-{1-[2-(methylsulfanyl)benzoyl]piperidin-3-yl}piperidin-4-yl)methanol
N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
4-(2,3-dihydro-1H-isoindole-2-carbonyl)-2,8-dimethylquinoline
N-{3-[4-(pyrimidin-2-yloxy)piperidine-1-carbonyl]phenyl}propanamide
4-(1-{4-[2-(cyclopentylmethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}-1-oxopropan-2-yl)-1,2-dihydrophthalazin-1-one
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-6-methoxy-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one