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5-{[4-(5-chloropyridin-2-yl)piperazin-1-yl]methyl}-2-cyclohexylpyrimidine
4-(2-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2-oxoethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(2-methoxyethyl)-1-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
2,2-bis(prop-2-en-1-yl)-1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
(3-benzyl-1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)methanol
N-[3-(4-methoxyphenyl)propyl]-6-[(thiolan-3-yl)amino]pyridine-3-carboxamide
5-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]pyridine-2-carbonitrile
N-[(5-methylfuran-2-yl)methyl]-4-(pyridin-2-yl)pyrimidin-2-amine
1-(5-phenyl-1,3,4-thiadiazol-2-yl)-N-[3-(pyridin-4-yl)propyl]piperidin-4-amine
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-1-methyl-3-phenyl-1H-pyrazole-5-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-N-{[7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
2-ethyl-4-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
5-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]-2,6-dimethyl-3,4-dihydropyrimidin-4-one
N-(2-methylpropyl)-1-[(1s,4s)-4-(dimethyl-1,2-oxazole-4-sulfonamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-{2-[(6-methyl-2-phenylpyrimidin-4-yl)amino]ethyl}imidazolidin-2-one
S-(4-fluoro-2-methylphenyl)-2-{1-oxa-8-azaspiro[4.5]decan-8-yl}-2-oxoethane-1-sulfonamido
3-[4-(1H-pyrazol-3-yl)piperidine-1-carbonyl]-1H-pyrazol-5-amine
1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-2-(2-hydroxyphenyl)ethan-1-one
[(1R)-1-(3-methoxyphenyl)ethyl]({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
3-{3-[4-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}-1H-indazole
2-(3,4-dimethoxyphenyl)-1-(7-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
7-cyclopentyl-2-(1H-imidazol-4-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
5-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
4-fluoro-N-(2-{[3-(4-hydroxyphenyl)-1H-pyrazol-5-yl]formamido}ethyl)benzamide
N-[2-(4-fluorophenyl)ethyl]-3-(2-phenylethyl)-1,2-oxazole-5-carboxamide
2-fluoro-N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-5-methylbenzene-1-sulfonamide
3-(2-fluorophenyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}pyrrolidine
1'-(3,5-difluoropyridine-2-carbonyl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
{imidazo[1,2-a]pyrimidin-6-ylmethyl}[3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amine
(1S,5R)-3-(3-chlorobenzoyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-4-(4-fluorophenyl)piperidin-4-ol
2-{5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
7-(diphenylmethyl)-2-oxa-7-azaspiro[4.5]decan-8-one
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-4-(4-methoxyphenyl)butane-1,4-dione
4-(2-{4-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-1H-pyrazol-1-yl}ethyl)morpholine
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
7-(propan-2-yl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-methyl-4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]-N-(quinolin-5-ylmethyl)benzamide
(4aS,8aS)-N-(3-cyanophenyl)-4a-hydroxy-decahydroisoquinoline-2-carboxamide
2-amino-6-(1-methylcyclopropyl)-4-[4-(1H-pyrazol-1-ylmethyl)phenyl]pyridine-3-carbonitrile
N-{4-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-1,2,3-triazol-4-yl]phenyl}acetamide
1-benzyl-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
(2S,4R)-N,N-diethyl-1-(3-hydroxypropanoyl)-4-(thiophene-2-amido)pyrrolidine-2-carboxamide
3-{2-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
3-{[3-methyl-1-(3-methylphenyl)-1H-1,2,4-triazol-5-yl]methoxy}pyridine
(1-{5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-3-yl)methanol
1-[1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea
N-(1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-1-oxopropan-2-yl)propanamide
N-(2-hydroxyethyl)-2-[(1-methyl-1H-indol-3-yl)sulfanyl]-N-(1,3-thiazol-2-ylmethyl)acetamide
8-benzyl-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione