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N-cyclobutyl-4-(thiomorpholine-4-sulfonyl)benzamide
3-[3-(3-methylthiophen-2-yl)phenyl]-1H-pyrazole
4-{[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}benzene-1-sulfonamide
N-{5H,6H,7H-cyclopenta[b]pyridin-7-yl}-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
3-{[(butan-2-yl)(pyridin-3-ylmethyl)amino]methyl}phenol
[(3R,4R)-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
7-(propan-2-yl)-N-(2,2,2-trifluoroethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
methyl 2-[3-(2-{[(2-chlorophenyl)methyl]carbamoyl}ethyl)piperidine-1-carbonyl]benzoate
4-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-2-[(4-methoxyphenyl)methyl]morpholine
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
3-(2-amino-1,3-thiazol-4-yl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
1-[2-methoxy-2-(thiophen-2-yl)ethyl]-5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazole
8-{2-[4-(hydroxymethyl)phenyl]acetyl}-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N3-(cyclohexylmethyl)-1-cyclopentyl-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1,3-benzoxazol-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
3-(1-methylpiperidin-3-yl)-1-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
7-(oxan-4-yl)-2-(pyridazine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-{[6-(3-ethoxyphenyl)pyridin-3-yl]methyl}morpholine
N-[2-(4-phenylpiperidin-1-yl)ethyl]pyrimidin-2-amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
3-(1-ethyl-1H-pyrazol-4-yl)-4-(3-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(2,6-dichlorophenyl)methyl]-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidine
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[4-(pyridin-4-yl)piperidin-1-yl]ethan-1-one
1-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]-N,N-dimethylazepan-4-amine
1-{3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]benzenesulfonyl}-4-methyl-1,2,3,6-tetrahydropyridine
3-ethyl-1-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)piperidine-3-carboxylic acid
4-(2,2-dimethylpropyl)-3-{2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
4-(4-fluoro-2-methylphenoxy)-1-(oxolan-3-ylmethyl)piperidine-4-carboxylic acid
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-2-(4-propanoylphenoxy)acetamide
N-(1-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenylpropanamide
5-(1H-imidazol-1-ylmethyl)-2-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)pyridine
(1R,2R,6S,7S)-N-(3-acetamido-4-fluorophenyl)-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
N-[2-(4-ethylmorpholin-2-yl)ethyl]-1H-indole-3-carboxamide
[(5-fluoro-3-methyl-1H-indol-2-yl)methyl](methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
1-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-5,5-diphenylpiperidin-2-one
(4S,4aS,8aS)-1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-phenyl-decahydroquinolin-4-ol
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1-(diphenylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-{4-[(dimethylsulfamoyl)amino]phenyl}-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}piperidin-4-amine
1-[2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)acetyl]-3-ethylpiperidine-3-carboxylic acid
2-{4-cyclobutyl-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-[2-(pyrrolidine-1-sulfonyl)ethyl]-1-(3-sulfamoylphenyl)urea
2-{1-cyclopentyl-4-[(2-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]morpholine
N-[(3-fluorophenyl)methyl]-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
methyl 4-{4-[2-(cyclopropylcarbamoyl)-5-methoxyphenoxy]piperidin-1-yl}pentanoate
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-propylpyrimidin-4-amine
4-{[3-(3-methylphenyl)piperidin-1-yl]methyl}pyridine
(3S,4S)-1-{1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]piperidin-4-yl}-4-(propan-2-yloxy)pyrrolidin-3-ol