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N-(cyclohex-1-en-1-ylmethyl)-4-propylpyrimidine-5-carboxamide
9-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
2-(4-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
1-[2-(2-ethoxyethoxy)phenyl]-3-[(1R,2S)-2-phenylcyclopropyl]urea
(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-4-(2-phenylethyl)piperidin-4-yl)methanol
3-(2-{5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-phenyl-1H-imidazol-1-yl}ethyl)-4-ethyl-4H-1,2,4-triazole
(1R,2S,9R)-11-[6-(methoxymethyl)pyrimidin-4-yl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
2-(3-fluorophenoxymethyl)-N-[(4-fluorophenyl)methyl]-N-methyl-1,3-oxazole-4-carboxamide
N-[4-(methylsulfanyl)phenyl]-3-[(3S,4R)-1-(pyridin-3-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
N-(1-methanesulfonylpiperidin-4-yl)-4-(piperidin-3-yl)benzamide
cyclopentyl 4-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)carbamoyl}amino)benzoate
1-(2-methoxyethyl)-2-oxo-3-(pyridin-3-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
N-[(4-hydroxyphenyl)methyl]-3-propyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
4-(4-methoxyphenoxymethyl)-1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidine
(3S,4S)-4-methyl-1-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]piperidine-3,4-diol
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-({[4-(propan-2-yl)phenyl]methyl}amino)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
4-{[2-(5-fluoro-2-methoxyphenyl)-1H-imidazol-1-yl](phenyl)methyl}pyridine
N-[1-(carbamoylmethyl)piperidin-4-yl]-4-hydroxy-2-phenylpyrimidine-5-carboxamide
4-(1H-imidazol-1-ylmethyl)-1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}piperidine
N-[2-(2-chloro-6-fluorophenyl)ethyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
1-(piperidin-1-yl)-2-[2-(trifluoromethyl)morpholin-4-yl]ethan-1-one
N-(2,3-dihydro-1H-inden-1-yl)-5-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
(3S,4R)-1-[3-(4-fluorophenoxy)propyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
(3R,9aR)-8-(2,5-difluorobenzoyl)-3-[(1S)-1-hydroxyethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(3S,4S)-4-hydroxy-1-(propan-2-yl)pyrrolidin-3-yl]-3-(3-hydroxy-3-methylbutyl)benzamide
4-(4-{[3-(2-hydroxyethyl)-4-(propan-2-yl)piperazin-1-yl]methyl}phenyl)but-3-yn-1-ol
2-[(2,6-dichlorophenyl)methyl]-N,N-diethyl-4-hydroxypyrimidine-5-carboxamide
(butan-2-yl)[(2-methyl-1H-imidazol-4-yl)methyl][(4-methylphenyl)methyl]amine
5-chloro-N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropylthiophene-2-sulfonamide
2-[3-(pyridin-3-yl)azetidin-1-yl]pyrimidin-4-amine
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}ethan-1-one
N-(1-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
9-methoxy-4-(5-methyl-1,2,4-oxadiazol-3-yl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
7-(1,3-benzothiazol-2-yl)-4-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(1,2-oxazolidin-2-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]propanamide
2-(5-amino-1,3,4-thiadiazol-2-yl)-1-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethan-1-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-3-ol
2-(pyridin-4-yl)-5-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazine-1-carbonyl}pyrimidine
2-methyl-9-(3-methyl-4-oxo-3,4-dihydroquinazoline-7-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(cyclohexylmethyl)-N-[2-(4-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
N-(1H-indazol-7-yl)-3-({methyl[1-methyl-1-(methylcarbamoyl)ethyl]amino}methyl)benzamide
2-{8-cyclopentyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-oxo-N-phenylacetamide
4-(carbamoylmethoxy)-N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]benzamide
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(4-fluoro-3-methylphenyl)ethan-1-one
2-methyl-6-({4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}methyl)pyridine
ethyl 4-[1-(3-methyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}propanamide