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1-[4-({7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)thiophen-2-yl]ethan-1-one
N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(5-methylthiophen-2-yl)ethyl]-3-(piperidin-3-yl)benzamide
2-[3-({[3-(azepan-1-yl)propyl](methyl)carbamoyl}amino)phenyl]-N-methylacetamide
N-[1-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
5-(1-cyclobutyl-1H-imidazol-2-yl)quinoline
5-phenyl-3-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]-1,2,4-oxadiazole
(2S,4R)-N-(1-benzothiophen-2-ylmethyl)-1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-N-methyl-4-(pyrimidin-2-ylsulfanyl)pyrrolidine-2-carboxamide
(3aR,6aR)-2-[(5-acetylthiophen-3-yl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-phenoxy-N-[(7-{[4-(propan-2-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]acetamide
ethyl 1-ethyl-5-(1H-indole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(cyclopropylmethyl)-N-methyl-5-[2-(4-methylphenoxy)acetyl]-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
2-fluoro-5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
4-{[4-(1-methyl-3-phenyl-1H-pyrazol-4-yl)-1H-1,2,3-triazol-1-yl]methyl}benzene-1-sulfonamide
3-{1-[(3-acetylphenyl)methyl]piperidin-3-yl}-N-(4-fluoro-2-methylphenyl)propanamide
7-methyl-2-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
2-amino-5-methyl-6-phenyl-4-(pyridin-4-yl)pyridine-3-carbonitrile
2-cyclopropyl-N-[2-(1H-indol-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
3-(1H-pyrazol-1-yl)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
5-cyclopropyl-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-N-[3-(pyridin-4-yl)propyl]-1H-pyrazole-4-carboxamide
N-cyclohexyl-1-methyl-3-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
(4S)-3-{2-[3-(2-fluorophenoxy)azetidin-1-yl]-2-oxoethyl}-4-(propan-2-yl)-1,3-oxazolidin-2-one
ethyl 3-(2-phenoxyethyl)-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidine-3-carboxylate
ethyl 4-(3-phenylpropyl)-1-(2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetyl)piperidine-4-carboxylate
3-{1-[(2-chlorophenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide
N-[(4-fluorophenyl)methyl]-N-(3-hydroxypropyl)-3,5,7-trimethyl-1H-indole-2-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(2S)-N-[3-(3-chlorophenyl)phenyl]-1-[1-(hydroxymethyl)cyclopropanecarbonyl]pyrrolidine-2-carboxamide
2-{2-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindole-1,3-dione
1-ethyl-4-{[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-3-methyl-1H-pyrazole
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-amine
(1S,5R)-6-(dimethyl-1,2-oxazole-4-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
8-(2,2-dimethylpropyl)-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[4-(butan-2-yloxy)-3-chlorophenyl]methyl}(methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
1-[3-(4H-1,2,4-triazol-4-yl)benzamido]-1,2,3,4-tetrahydronaphthalene-1-carboxylic acid
N-benzyl-6-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
4-[(2S)-1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]pyrrolidine-2-carbonyl]morpholine
4-(4-ethoxy-3-methylphenyl)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]butan-1-one
1-acetyl-N-[2-(3-propoxyphenyl)ethyl]piperidine-3-carboxamide
2-[3-(propan-2-yloxy)phenyl]-6-(pyrrolidine-1-carbonyl)pyrazine
8-[(2-chlorophenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-benzyl-5-(4-ethoxybenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine
8-[2-(2-hydroxyethoxy)ethyl]-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
4-[1-(1-cyclopropylethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-5-methyl-2-(thiophen-2-yl)-1,3-oxazole
3-[(3-chlorophenyl)methyl]-N-[(4-phenyloxan-4-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
2-{[4-(2,3-dichlorophenyl)piperazin-1-yl]methyl}pyridine-3-carboxylic acid