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1-cyclohexyl-4-[3-(1H-pyrazol-1-yl)propanoyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
1-(3-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pentan-1-one
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[(5-methylthiophen-2-yl)methyl]benzamide
methyl 2-{2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-methylacetamido}acetate
3-[1-(2-amino-3-cyclopentylpropanoyl)piperidin-4-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{[1-(2,6-dimethoxypyrimidin-4-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
1-[(3-fluorophenyl)methyl]-4-[3-(methylsulfanyl)propyl]piperazin-2-one
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-[1-(4-fluorophenyl)propan-2-yl]-1,4-diazepan-5-one
({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[(2-phenyl-1,3-thiazol-4-yl)methyl]amine
4-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-[2-(dimethylamino)ethyl]pyrrolidin-2-one
methyl 4-[({2-[1-(adamantan-2-ylmethyl)-5-oxopyrrolidin-2-yl]ethyl}amino)methyl]benzoate
6-[(3-methoxyphenyl)methoxy]-4-[2-(methylsulfanyl)acetyl]-1-(2-phenylethyl)-1,4-diazepan-2-one
N,2-dimethyl-6-(piperidin-3-yl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidin-4-amine
N-methyl-N-[1-(4-methylquinazolin-2-yl)pyrrolidin-3-yl]acetamide
N-{3-[(5-methylpyridin-2-yl)amino]propyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-ethyl-4-[(4-methyl-1H-imidazol-5-yl)methyl]-1-(propan-2-yl)piperazine
3-(piperidin-1-ylmethyl)-1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine
N-(furan-2-ylmethyl)-5-methyl-4-{[2-(piperidin-1-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-({7-[2-(cyclohex-1-en-1-yl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1H-indole-2-carboxamide
1-methyl-8-(2-methylpyridin-4-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-N-butyl-5-cyclopropyl-N-methyl-1H-pyrazole-4-carboxamide
N-{[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
methyl 8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-3,5-dimethyl-1H-indole
2-{[(1,3-benzothiazol-2-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
4-cyclobutanecarbonyl-7-(6,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(3,4-dimethoxyphenyl)methyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-(pyridin-4-ylmethyl)acetamide
3-(3-hydroxyquinoxalin-2-yl)-N-[(5-methylpyrazin-2-yl)methyl]propanamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[3-(propan-2-yloxy)propyl]piperidin-2-one
[(3,5-dimethoxyphenyl)methyl](methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
5-(1-cyclohexanecarbonylpiperidin-4-yl)-3-[3-(dimethylamino)propyl]-5-[(2-methylphenyl)methyl]imidazolidine-2,4-dione
2-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
2-[2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-8-methyl-2,8-diazaspiro[5.5]undecane
2-methyl-4-{3-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]phenyl}but-3-yn-2-ol
3-[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]-N-(1,3-thiazol-2-yl)propanamide
3-chloro-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-6-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide
3-cyclopropyl-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}propanamide
[2-(4,6-dimethylpyrimidin-2-yl)ethyl]({[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl})amine
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
3-(1-methyl-1H-pyrazol-4-yl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-ethyl-N-[2-(4-fluorobenzenesulfonyl)ethyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}ethan-1-one
2-(2-ethoxyphenyl)-2-[methyl(oxan-4-ylmethyl)amino]acetic acid
2,5-dimethyl-3-(3-{1-[(4-methyl-1,3-thiazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrazine
1-[(3-fluorophenyl)methyl]-N-methyl-N-(1,2-oxazol-5-ylmethyl)-6-oxopiperidine-3-carboxamide
(1S,3R)-N,2,2,3-tetramethyl-3-[3-(2-methylphenoxy)azetidine-1-carbonyl]cyclopentane-1-carboxamide
1-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-3-phenoxypropan-1-one
4-[(dimethylamino)methyl]-N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide
N-[2-(dimethylamino)ethyl]-N-(oxolan-2-ylmethyl)-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide