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N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-5-(thiophen-3-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[3-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-6-methylpyridine
methyl 4-[(10-{[1-(furan-2-yl)ethyl]carbamoyl}-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-3-yl)methyl]benzoate
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-methyl-2-oxoimidazolidine-4-carboxamide
methyl 9-(cyclopentyloxy)-3-[(3,4-dimethylphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(2-{4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl}ethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
7-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-{2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-1H-1,2,4-triazol-5-yl]ethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
4-chloro-2-({3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
1-[2-(3-methoxyphenoxy)ethyl]-4-(oxane-2-carbonyl)piperazine
2-(1H-imidazol-2-yl)-N-(6-methylpyridin-3-yl)benzamide
2-(4-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)-N,N-dimethylacetamide
(oxolan-2-ylmethyl)(pyridin-2-ylmethyl){[3-(pyrimidin-2-yloxy)phenyl]methyl}amine
{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
8-(3-ethoxypropanoyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(3-cyclopentylpropyl)-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamide
1-(4-{5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-diazepan-1-yl)ethan-1-one
8-[(4-hydroxyphenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-hydroxy-N-methyl-2-(4-methylphenyl)-N-[1-(1,3-thiazol-2-yl)ethyl]pyrimidine-5-carboxamide
2-(1-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-2-yl)-1,3-thiazole
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-(5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperidine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
2-methyl-6-{[(1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)amino]methyl}pyrimidin-4-ol
3-(2-methoxyethyl)-1-[6-(methoxymethyl)pyrimidin-4-yl]piperidine-3-carboxylic acid
(3R,4R)-4-amino-1-{5-[(4-methylpiperazin-1-yl)methyl]furan-2-carbonyl}piperidin-3-ol
2-{[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]amino}-N-(pyrazin-2-yl)acetamide
N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-3-propyl-1H-pyrazole-5-carboxamide
1-{2-methyl-5-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]phenyl}imidazolidin-2-one
3-(1,3-benzothiazol-2-yl)-N-benzylpiperidine-1-sulfonamide
(2-{4-[6-(methoxymethyl)pyrimidin-4-yl]morpholin-2-yl}ethyl)dimethylamine
(1R,2R)-2-{[(8-chloroquinolin-2-yl)methyl](ethyl)amino}cyclohexan-1-ol
3-(oxolan-3-yl)-5-(4,5,6,7-tetrahydro-2-benzothiophen-1-yl)-1,2,4-oxadiazole
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-6-(1-propyl-1H-1,2,3-benzotriazol-5-yl)pyridine-3-carbonitrile
N-[4-(3-methylpiperidine-1-carbonyl)phenyl]-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
N-{2-[benzyl(methyl)amino]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl}-2-acetamidoacetamide
1-(dimethyl-1,3-oxazole-5-carbonyl)-3-phenylpiperazine
1-[2-methoxy-5-({[2-(2-methylphenyl)ethyl]amino}methyl)phenoxy]-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
2-(2-hydroxyethyl)-8-[3-(4-methoxyphenyl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
(3S,4R)-4-phenyl-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidine-3-carboxylic acid
1-{4-[(1R,3S,4S)-3-hydroxy-4,7,7-trimethylbicyclo[2.2.1]heptane-1-carbonyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
N-(3-fluorophenyl)-3-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanamide
N-[4-(2-fluorophenoxy)phenyl]-1-(furan-2-carbonyl)piperidine-4-carboxamide
2-(methylsulfanyl)-5-[4-(pyridin-4-yl)piperidine-1-carbonyl]pyrimidine
N-cyclopropyl-5-(1,2,3,4-tetrahydroquinoline-8-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[1-(4-{4-[hydroxy(phenyl)methyl]piperidine-1-carbonyl}phenyl)-1H-pyrazol-4-yl]oxane-4-carboxamide
4-[6-amino-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-2-chlorobenzamide
N-({5-[(3,4-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
1-(2-hydroxyethyl)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1H-1,3-benzodiazole-5-carboxamide
2-({[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)propanamide