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N-{1-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
8-(5-propylthiophene-3-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-methyl-N-(thiophen-3-ylmethyl)quinoline-2-carboxamide
N-(3-chloro-4-ethoxyphenyl)-3-(pyrrolidine-1-carbonyl)piperidine-1-carboxamide
3,5-dimethyl-N-(4-pentanamidophenyl)-1H-pyrazole-4-carboxamide
2-(3-fluorophenyl)-1-{4-[2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
2-cyclohexyl-5-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]pyrimidine
2-(oxolan-2-ylmethoxy)-1-[4-(2-phenylethyl)piperidin-1-yl]ethan-1-one
1-[2-(4-chloro-2-methylphenoxy)ethyl]-4-(oxolane-3-carbonyl)piperazine
5-(2,6-difluorophenoxymethyl)-N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-1,2-oxazole-3-carboxamide
2-methyl-N-[(7-{[4-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]butanamide
methyl 5-[(4-hydroxy-4-methylpentan-2-yl)amino]-3-(2-methoxyacetamido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-[4-(methoxymethyl)-5-methyl-1,2-oxazol-3-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-(2-{4-[(4-phenylpiperidin-1-yl)methyl]phenoxy}propyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(2H-indazol-2-yl)acetamide
methyl 4-[(2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}phenyl)formamido]butanoate
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
2-[4-({8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-3-methyl-1H-pyrazol-1-yl]ethan-1-ol
1-{2-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]piperidin-1-yl}pent-4-en-1-one
2-{[(3R,5S)-1-[(2,4-difluorophenyl)methyl]-5-(4-methyl-1,4-diazepane-1-carbonyl)pyrrolidin-3-yl]sulfanyl}-1H-1,3-benzodiazole
N-cyclopropyl-N-{[4-(methylsulfanyl)phenyl]methyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-benzyl-N,N-dimethyl-5-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(4-benzyl-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)methanol
N-[2-(2-chlorophenyl)-2-hydroxyethyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]benzene-1-sulfonamide
N-[(4-methyl-1,4-oxazepan-6-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
4-{imidazo[1,2-a]pyridine-2-carbonyl}-1-(3-methoxyphenyl)piperazin-2-one
2-[(2-methylprop-2-en-1-yl)oxy]-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
[(1-cyclohexylpiperidin-3-yl)methyl](1,2-oxazol-3-ylmethyl)(pyridin-3-ylmethyl)amine
[1-(4-chlorophenyl)propan-2-yl][1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]amine
(1R,5R)-3-(2,3-dihydro-1H-indene-5-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-(1H-indol-5-ylmethyl)propanamide
methyl 2-{[5-(1H-1,3-benzodiazol-1-ylmethyl)-1H-pyrazol-3-yl]formamido}pentanoate
N-ethyl-3-(2-methyl-1H-imidazol-1-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide
N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-sulfamoylbenzamide
(2-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-4-yl)methanol
methyl (2S)-3-methyl-2-({5-[(quinolin-6-yloxy)methyl]-1,2-oxazol-3-yl}formamido)butanoate
N-methyl-N-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-2-(3-methylphenyl)ethan-1-one
(3R,4S)-1-[3-(azepan-1-ylmethyl)benzoyl]-4-phenylpyrrolidin-3-amine
5-[2-(1-ethylpiperidin-4-yl)acetyl]-N,N-dimethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-2-(methylamino)-1,3-thiazole-4-carboxamide
1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-1-(furan-2-ylmethyl)piperidine-3-carboxamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
6-(difluoromethyl)-2-(4-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}phenyl)-3,4-dihydropyrimidin-4-one
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(5,6-dimethylpyrazin-2-yl)pyrrolidin-3-yl]methanol
1-(1-methylpiperidin-4-yl)-N-(prop-2-en-1-yl)piperidine-3-carboxamide
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-(1,3-thiazol-2-ylmethyl)-decahydroisoquinoline