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N-[1-(4-fluorophenyl)-2-hydroxyethyl]-3-(pyridin-4-yl)propanamide
4-[1-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-4-phenyl-1H-imidazol-5-yl]pyridine
(1S,5R)-6-benzyl-3-[(3-hydroxy-4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{4-[(cyclobutylamino)methyl]-2-methoxyphenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
methyl 1-[(3R,5S)-1-[(4-ethylphenyl)methyl]-5-[(thiophen-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
4-acetyl-N-{[2-(dimethylamino)pyridin-3-yl]methyl}benzene-1-sulfonamide
N-(1-{7-[(3-chlorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclopropanecarboxamide
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-2-(2-oxopiperidin-1-yl)acetamide
N-[(3S,4R)-1-[2-(methylsulfanyl)pyridine-3-carbonyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
N-[2-(4-methylmorpholin-2-yl)ethyl]-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)acetamide
2-amino-4-[2-(furan-2-yl)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
6-oxo-1-(3-phenylpropyl)-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
N-methyl-4-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]pyridin-2-amine
N-methyl-N-(prop-2-en-1-yl)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-methoxy-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,2-oxazolidine
1-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}-4-(cyclopropylmethyl)piperazine
7-[2-(piperidin-1-yl)acetyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4,6,7-trimethyl-2-[4-(quinolin-6-ylmethyl)-1,4-diazepan-1-yl]quinazoline
methyl 3-[2-(2-methoxyphenyl)acetyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[1-(3-hydroxyadamantan-1-yl)ethyl]-5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-methyl-6-oxo-4-(4-phenyl-1,3-thiazol-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
2-chloro-N-{2-[2-(4-methylphenyl)-1H-imidazol-1-yl]ethyl}benzamide
N-cyclopropyl-1-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
3-methyl-1-[1-(6-{[(1r,4r)-4-hydroxycyclohexyl]amino}pyridine-3-carbonyl)piperidin-3-yl]butan-1-one
3-(1-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-chlorophenyl)urea
4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-methylphenyl)methyl]piperidine
N-[(5-chlorothiophen-2-yl)methyl]-1-[2-(dimethylamino)ethyl]-6-oxopiperidine-3-carboxamide
6-{methyl[(3-methyl-1H-pyrazol-4-yl)methyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
5-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-(2-methylpropyl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-3-(1,3-dimethyl-4-phenyl-1H-pyrazol-5-yl)urea
2-(3-methoxyphenyl)-1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
3-(2-oxopyrrolidin-1-yl)-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)propanamide
ethyl 1-[(4-methoxyphenyl)methyl]-5-(1,3-thiazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(1R,5R)-6-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
2-(5-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyrazine
1-[1-(2,4-dimethylphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-2-methylpropan-1-ol
1-(1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)piperidin-4-ol
4-(hydroxymethyl)-1-[1-(4-phenoxyphenyl)-1H-1,2,3,4-tetrazol-5-yl]azepan-4-ol
1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-3-(3-methoxyphenyl)propan-1-one
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
1-benzyl-5-methanesulfonamido-N-[(3-methoxyphenyl)methyl]-2-methyl-1H-1,3-benzodiazole-7-carboxamide
4-hydroxy-2-[(phenylsulfanyl)methyl]-N-[2-(1,3-thiazol-2-yl)ethyl]pyrimidine-5-carboxamide
3-[1-(1-cyclopropyl-1H-pyrrol-2-yl)-N-(2-phenylethyl)formamido]propanamide
5-[1-(4-chlorobenzoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
1-[2-methyl-4-(4-methylphenyl)-5-oxopiperazin-1-yl]propane-1,2-dione
N,N-diethyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
methyl (1S,3S,3aR,6aS)-1-(hydroxymethyl)-5-methyl-3-(5-methyl-1-propyl-1H-pyrazol-4-yl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-4-methoxybenzamide