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N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
(2R)-1-{2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carbonyl}pyrrolidine-2-carboxamide
(1,4-dioxan-2-ylmethyl)(methyl){[3-(1H-pyrazol-4-yl)phenyl]methyl}amine
N-ethyl-1-[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]pyrrolidine-3-carboxamide
4-[2-hydroxy-4-(methylsulfanyl)butanoyl]-1-(2-methoxyphenyl)piperazin-2-one
1-(4-cyano-2-ethylphenyl)-3-(2-methanesulfonamidoethyl)urea
2-[(1-methylpiperidin-4-yl)methyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(1S,6R)-3-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
(1R,3S)-7-[(3-chloro-2-fluorophenyl)methyl]-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
3-methyl-1-(2-methylpropyl)-8-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-1-phenyl-1H-1,2,3-triazole-5-carboxamide
3-[methyl({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amino]propane-1,2-diol
4-(2,6-dimethylpyridin-3-yl)-N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]pyrimidin-2-amine
3-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]acetamide
methyl 9-(oxan-2-ylmethoxy)-7-oxo-3-[(4-oxo-4H-chromen-3-yl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N,N-dimethyl-4-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}aniline
ethyl 2-(1-{1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-2-yl)acetate
1-cyclopentyl-N3-methyl-N3-(2-methylpropyl)-4-oxo-N5-{[2-(trifluoromethyl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
2-{[4-(adamantan-1-yl)piperazin-1-yl]methyl}benzoic acid
(5S,9aS,9bS)-5-[5-(methoxymethyl)furan-2-yl]-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-methyl-1-[(4-phenoxyphenyl)methyl]-1,4-diazepan-5-one
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
3-(2-{3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-oxoethyl)-4-(3-methylbutyl)piperazin-2-one
N-[2-fluoro-5-({[3-(4-methylpiperazin-1-yl)propyl]carbamoyl}amino)phenyl]-2-methylpropanamide
propan-2-yl 2-(3-methoxyphenyl)pyrrolidine-1-carboxylate
4-{1-[(2,4-difluorophenyl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
4-{[4-(carbamoylmethoxy)-3-chlorophenyl]methyl}-N-cyclopropylpiperazine-2-carboxamide
1-[3-(2,3-dihydro-1H-isoindol-2-ylmethyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
N-[2-(3-fluorophenyl)ethyl]-4-[(3-methoxypropyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-methoxy-2-phenyl-N-(1-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
N-ethyl-3-(4-hydroxyphenyl)-N-(oxan-2-ylmethyl)benzamide
2-{[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-3-methylquinoxaline
(1H-1,3-benzodiazol-2-ylmethyl)(ethyl)({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)amine
9-[2-(4-fluorophenoxy)ethyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
4-[(1-phenylmethanesulfonylpyrrolidin-3-yl)methyl]benzoic acid
2-{2-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
N-[(2-chlorophenyl)methyl]-3-[1-(3-fluoro-4-methoxybenzoyl)piperidin-3-yl]propanamide
2-{4-[(3,5-difluorophenyl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
methyl[(5-methylthiophen-2-yl)methyl]{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-3-acetamidopropanamide
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[4-(trifluoromethyl)benzoyl]piperidine
3-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}piperidine-1-carboxamide
{1-[2-(methylsulfanyl)pyridine-3-carbonyl]-3-(2-phenoxyethyl)piperidin-3-yl}methanol
6-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
2-(ethoxymethyl)-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-cyclopropyl-5-(3-phenylpiperazine-1-carbonyl)pyrimidine
1-(cyclohexylmethyl)-6-oxo-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]piperidine-3-carboxamide