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3-[2-(2-methylphenyl)ethyl]-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidine
3-cyclobutyl-4-(1-propyl-1H-imidazol-2-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(5S,9aS,9bS)-5-(2,1,3-benzoxadiazol-4-yl)-2-cyclopentyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-methoxy-6-(3,4,5-trifluorophenyl)pyridazine
2-(1-{1-[1-(trifluoromethyl)cyclopropanecarbonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-amine
2-amino-4-{3-[(dimethylamino)methyl]phenyl}-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-methyl-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
N-(isoquinolin-1-yl)-4-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}benzamide
methyl 3-[(1-methyl-1H-indol-3-yl)methyl]-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methylthiophen-2-yl)methyl]acetamide
1-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}-2-(pyridin-4-yl)ethan-1-one
(3aR,6aR)-2-(2-chloro-5-methylbenzoyl)-5-(cyclobutylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{[({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}-4-methoxyphenol
4-(2,4-dichlorophenyl)-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(3R,4S)-1-(2-methoxyethyl)-4-propylpyrrolidin-3-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carboxamide
2-[1-(1-cycloheptylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
5-{[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
6-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
5-methanesulfonyl-N,2-dimethyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-4-amine
4-{3-[4-(dimethylamino)azepane-1-carbonyl]phenyl}-2-methylbutan-2-ol
(1-{2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}pyrrolidin-3-yl)methanol
5-{[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]methyl}-2,1,3-benzoxadiazole
(3aR,6aS)-1-oxo-5-{[1-(prop-2-en-1-yl)-1H-1,3-benzodiazol-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1,9-dimethyl-4-({2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}methyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidine-4-carboxylic acid
methyl 4-methoxy-3-[({[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}carbamoyl)amino]benzoate
1-(azepan-1-yl)-3-[4-chloro-2-({[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
3-[(4-fluorophenyl)methyl]-5-{1-[2-(2-methoxyphenoxy)acetyl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
3-({[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]amino}methyl)-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-(4-methoxyphenyl)-6,6-dimethyl-4-[5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carbonyl]piperazin-2-one
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-[(3,5-difluorophenyl)methyl]-8-(5,6-dimethylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-1-(thiomorpholin-4-yl)ethan-1-one
6-(4-aminopyridin-3-yl)-2,3,4,9-tetrahydro-1H-carbazol-1-one
methyl 4-({3-[2-(furan-3-ylformamido)ethyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)benzoate
1-ethyl-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazole
6-[4-(2-methoxyethyl)piperazine-1-carbonyl]-N-[2-(2-methoxyphenyl)ethyl]-5-methylthieno[2,3-d]pyrimidin-4-amine
1-(4-phenylpiperazin-1-yl)-3-[1-(thian-4-yl)piperidin-4-yl]propan-1-one
4-(cyclopropylmethyl)-1-(2-methylpyrimidin-4-yl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-[(1-cyclohexylpiperidin-3-yl)methyl]-N-(pyridin-3-ylmethyl)-4H-thieno[3,2-b]pyrrole-5-carboxamide
1-ethyl-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1H-pyrazole-5-carboxamide
(4aS,8aS)-2-cyclobutanecarbonyl-7-(3-methyl-1,2-oxazole-5-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-5-methoxyfuran-2-carboxamide
5-(2,3-dihydro-1,4-benzodioxine-6-sulfonyl)-3-propyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
(5S)-5-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidine-1-carbonyl]pyrrolidin-2-one
1-(2-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-2-oxoethyl)piperidin-2-one
N-[(3-methylphenyl)methyl]-N-(propan-2-yl)thiophene-2-carboxamide
N-{1-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}-3-(2-methyl-1H-indol-1-yl)propanamide