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[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl](methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(3-methoxyphenyl)methyl]methylamine
1-(4-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
5-(2-fluorophenyl)-N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,2,4-triazin-3-amine
N-(2,2-difluoroethyl)-5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
methyl (2S)-1-[(4-{[4-(difluoromethoxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]pyrrolidine-2-carboxylate
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(morpholin-4-yl)-6-(thiophen-3-yl)pyridine-3-carboxamide
4-[(4-fluorophenyl)methyl]-11-({[3-(trifluoromethyl)phenyl]methyl}amino)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-benzyl-N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-{2-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-oxoethyl}imidazolidine-2,4-dione
methyl (2S,4R)-1-methyl-4-{9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-amido}pyrrolidine-2-carboxylate
4-methoxy-1-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidine
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidine-3-carbonitrile
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-(methoxymethyl)piperidine-1-sulfonamide
(1S,5R)-3-{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonane
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2-propylpyridine-4-carboxamide
({3-[(dimethylamino)methyl]phenyl}methyl)[(2-ethylpyrimidin-5-yl)methyl]methylamine
5-[(6-chloropyridin-3-yl)methyl]-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-{10-azabicyclo[4.3.1]decane-10-carbonyl}-8-methyl-2-(pyrimidin-5-yl)quinoline
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)acetamide
1-[1-(2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzoyl)piperidin-3-yl]-3-methylbutan-1-one
1-[4-({[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl)amino}methyl)thiophen-2-yl]ethan-1-one
2-{4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
9-methyl-3-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}-3,9-diazaspiro[5.6]dodecan-10-one
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2,2-dimethylpropan-1-one
2-(2-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}phenyl)-6-methyl-3,4-dihydropyrimidin-4-one
2-(2-chloro-4-fluorophenoxymethyl)-N-(2-methoxyethyl)-1,3-oxazole-4-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(furan-2-ylmethyl)acetamide
N-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-(2-chlorophenyl)-3-{1-[1-(3-hydroxy-2,2-dimethylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
3,5-dimethyl-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)-1,2-oxazole-4-sulfonamide
4-[({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]hepta-1,6-dien-4-ol
5-{[(4aS,7aR)-4-benzyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
4-(butan-2-yl)-3-[(4-hydroxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2,3-dihydro-1H-inden-5-yl)-3-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]urea
N-(1-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylpyridine-2-carboxamide
3-(2-chlorophenyl)-6-(furan-3-ylmethyl)-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
5-{1-[2-(3-fluorophenyl)acetyl]piperidin-4-yl}-5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]-N-[2-(1H-indol-1-yl)ethyl]piperidin-4-amine
5-(methoxymethyl)-N-(2-phenylethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(propan-2-yloxy)propanamide
4-ethyl-3-{1-[2-(1H-indol-3-yl)acetyl]piperidin-3-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(3-hydroxypropyl)-2-[1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
[1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-3-[(4-fluorophenyl)methyl]piperidin-3-yl]methanol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methylmorpholine-2-carboxamide
1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(2-methylphenoxymethyl)piperidine
3-fluoro-N-(1-{1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-(1-{1-[2-(propan-2-yloxy)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](1H-indol-3-ylmethyl)(2-methoxyethyl)amine