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3-(3,4-dimethylphenyl)-N-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}propanamide
N-(1-benzofuran-2-ylmethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
N-[1-(hydroxymethyl)cyclopentyl]-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-methyl-4-{3-methyl-5-[3-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazol-1-yl}-1,2-dihydroquinolin-2-one
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H-pyrazole-4-carboxamide
8-[1-(4-chlorophenyl)cyclobutanecarbonyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
4-[3-(4-fluorophenyl)benzoyl]-7-{[3-(methoxymethyl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
[(3S,5R)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
2-(2-methoxyethyl)-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-1,3-benzoxazole-6-carboxamide
2-[5-(2-cyclopropylpyrimidin-5-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl]acetamide
N-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1-methanesulfonylpiperidin-4-amine
1-(2-chloroprop-2-en-1-yl)-3-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-3-(1H-pyrazol-1-yl)benzamide
{7-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]-5-fluoro-2,3-dihydro-1-benzofuran-2-yl}methanamine
3-(3-fluorophenyl)-1-[2-(piperidin-1-yl)ethyl]-6-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
N-(cyclopropylmethyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-4-(piperidin-3-yl)benzamide
2-{4-[1-(3-methylpyridin-2-yl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
3-{[1-(2-amino-2-methylpropyl)pyrrolidin-3-yl]methyl}benzoic acid
(3R,4R)-1-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-3-methyl-4-(oxan-4-yl)piperidin-4-ol
5-acetamido-2-ethyl-N-[2-(furan-2-yl)ethyl]-1-(pyridin-3-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}(methyl)[1-(pyridin-2-yl)ethyl]amine
(5S,9aS,9bS)-2-cyclopentyl-5-(3-ethoxy-4-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(oxolan-3-ylmethyl)-4-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidine
(1R,5S,6S)-6-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-3-azabicyclo[3.1.0]hexane
1-(2-{2-benzyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)imidazolidine-2,4-dione
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-(pyrrolidin-1-yl)piperidin-3-yl]-1-[4-(2-methylphenyl)piperazin-1-yl]propan-1-one
N-[3-(azepan-1-yl)propyl]-1-[(2-fluorophenyl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
methyl[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
(2S)-1-(4-{[(3-methoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)pyrrolidine-2-carboxamide
5-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-5-[(3-methoxyphenyl)methyl]-3-methylimidazolidine-2,4-dione
6-({5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-2-methyl-2,3-dihydropyridazin-3-one
1-(4-fluorophenyl)-4-{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}piperazine
1-amino-N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)cyclopropane-1-carboxamide
6-(2-chlorophenyl)-N-(2-methoxyethyl)-N,7-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-[(3-methoxyphenyl)methyl]-8-(pent-2-yn-1-yl)-2,8-diazaspiro[4.5]decan-3-one
5,7-dimethyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]pyrido[2,3-d]pyrimidin-4-amine
N-[2-hydroxy-2-(pyridin-3-yl)ethyl]-2,7,8-trimethylquinoline-4-carboxamide
5-benzyl-5-{1-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]piperidin-4-yl}imidazolidine-2,4-dione
2-[(4aR,8aR)-7-cyclobutanecarbonyl-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-N-(1,3-dimethyl-1H-pyrazol-4-yl)acetamide
3-{2-[7-(1-hydroxy-3-phenylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
9-(2H-1,3-benzodioxol-5-ylmethyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-1H-indole-6-carboxamide
4-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)thiomorpholine
2-methyl-2-(2-{[(1S)-1-(3-methylpyridin-2-yl)ethyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)propanoic acid
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(2,4-difluorophenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[3-(2-methoxyethyl)-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl]-3-methylpiperidine
(2S)-1-(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)pyrrolidine-2-carboxamide
(4aR,7aS)-1-acetyl-4-(pyridazine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione