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(3S,4S)-1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
N-methyl-2-[(propan-2-yl)amino]-N-[1-(pyridin-3-yl)propyl]pyrimidine-5-carboxamide
1-{4-phenyl-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}ethan-1-one
5-[1-(2-methoxy-2-phenylacetyl)piperidin-4-yl]-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-benzoyl-N-methyl-N-[2-(2-methylpiperidin-1-yl)ethyl]piperidin-4-amine
6-methyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-(3-phenylpropyl)-11-{[2-(pyridin-3-yl)ethyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-2-amine
1-(morpholin-4-yl)-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(4-chlorophenyl)methyl]-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
(3S,9aR)-8-[(3-chlorophenyl)methyl]-3-[(4-hydroxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-({5-[(4-cyanophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
3-(1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)benzoic acid
1-(4-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-1,4-diazepan-1-yl)-2-methoxyethan-1-one
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2,2,3,3-tetramethylcyclopropane-1-carboxamide
2-(2-chlorophenoxy)-1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
3-({cyclohexyl[(3-methylphenyl)methyl]amino}methyl)pyrrolidin-3-ol
7-(cyclopropylmethyl)-2-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)(3-methylbut-2-en-1-yl)amine
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
2-(2-{[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}ethyl)-6-phenyl-2,3-dihydropyridazin-3-one
N-[2-(2-chlorophenyl)ethyl]-3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
5-(4-acetylphenoxymethyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,2-oxazole-3-carboxamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
4-(1H-imidazol-2-yl)-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)piperidine
2-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)-4-hydroxyquinoline-6-carboxamide
(4aS,8aR)-6-(2-fluorobenzoyl)-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
4-(3-{4-azaspiro[2.5]octane-4-carbonyl}phenyl)-2-methylbutan-2-ol
(3S,4R)-1-(2-amino-2-methylpropyl)-4-(2H-1,3-benzodioxol-5-yl)pyrrolidine-3-carboxylic acid
3-[(4-ethyl-5-methylpyrimidin-2-yl)amino]-2-(thiophen-3-ylmethyl)propan-1-ol
N,7,8-trimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[(1-methylpyrrolidin-2-yl)methyl]quinoline-4-carboxamide
1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-3-{[5-(pyridin-4-yl)-1,3,4-oxadiazol-2-yl]sulfanyl}propan-1-one
2-(pyridin-3-yloxy)-N-[1-(pyrrolidin-1-ylmethyl)cyclohexyl]acetamide
2-[(2,3-difluorophenyl)methyl]-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
6-(2-chlorophenyl)-7-(3-methylbut-2-en-1-yl)-2-(pyrrolidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
[(3R,4R)-1-(5-chlorofuran-2-carbonyl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
ethyl 2-[(5-{2-amino-6-oxo-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-8-yl}pyrimidin-2-yl)(methyl)amino]acetate
N-[4-(ethylcarbamoyl)-2-methylphenyl]-3-[(2-methylphenyl)methoxy]azetidine-1-carboxamide
2-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-4-carboxamide
2-ethyl-5-[4-(oxan-4-yl)piperazine-1-carbonyl]pyrimidine
1-[(3-fluorophenyl)methyl]-6-oxo-N-{[3-(trifluoromethoxy)phenyl]methyl}piperidine-3-carboxamide
1-(2-{4-[(2,4-dimethoxyphenyl)methyl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
1-(4-{[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]methyl}phenyl)imidazolidin-2-one
N-[(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidin-3-yl)methyl]-1H-pyrrole-2-carboxamide
N-ethyl-5-(4-methoxy-4-phenylpiperidine-1-carbonyl)pyrimidin-2-amine
1-{1-[(2-chlorophenyl)methyl]piperidin-4-yl}-N-(2-hydroxyethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[3-(dimethylamino)phenyl]-3-(2-methylpiperidin-1-yl)azetidine-1-carboxamide