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(1R,5R)-N,N-dimethyl-6-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-[(5-methyl-1H-pyrazol-3-yl)methyl]-4-[4-(4-methylphenyl)-1H-1,2,3-triazol-1-yl]piperidine
2-(3-phenyl-1H-1,2,4-triazol-5-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
8-(isoquinoline-3-carbonyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[2-methoxy-1-(pyridin-2-yl)ethyl]-3-methyl-1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}urea
7-methoxy-3-[(3-methoxypiperidin-1-yl)methyl]-2-(3-methylphenyl)quinoline
N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}thieno[2,3-d]pyrimidin-4-amine
1-(2-methoxyethyl)-8-[(4-methoxyphenyl)methyl]-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 2-cyclohexyl-3-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-3-oxopropanoate
1-cyclohexyl-N-methyl-N-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-hydroxy-1-(2-methoxyethyl)-3-({4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)piperidin-2-one
{1-[2-(morpholin-4-yl)benzoyl]-3-(2-phenoxyethyl)piperidin-3-yl}methanol
1-(1,3-dimethyl-1H-indole-2-carbonyl)azetidin-3-ol
5-[(3-fluorophenyl)methyl]-5-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-3-(2-methylpropyl)imidazolidine-2,4-dione
3-[(3R,4S)-4-(dimethylamino)-1-[(5-methylthiophen-2-yl)sulfonyl]piperidin-3-yl]propanoic acid
1-[2-(methylsulfanyl)benzoyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
(1S,5R)-3-[2-(benzyloxy)ethyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-methoxyethyl)-N-[(3-methylthiophen-2-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperidin-3-ol
1-[7-(5-chloro-2-methoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
2-methyl-4-{4-[2-(pyridin-2-yl)piperidine-1-carbonyl]phenyl}butan-2-ol
3,3-dimethyl-N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]butanamide
4-({1-benzyl-5-[2-(5-methyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,4-triazol-3-yl}methyl)-1-methylpiperidine
N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]-3-[(4-fluorophenyl)formamido]propanamide
5-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
4-(2-fluorophenoxy)-1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperidine
1-{2-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
3-(3-acetylphenyl)-1-(3-methylbut-2-en-1-yl)-6-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
4-(3-fluorobenzoyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(4-methoxy-3,5-dimethylphenyl)-1-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]urea
2,3-dimethoxy-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
2-(methylsulfanyl)-6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
N,N-dimethyl-1-{5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-3-amine
ethyl 4-(1-oxo-1,2,3,4-tetrahydroisoquinoline-3-amido)piperidine-1-carboxylate
N-{2-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-3-yl]ethyl}methanesulfonamide
7-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-4-[4-(methylsulfanyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
2-methyl-4-[1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-3-yl]-6-(pyrrolidin-1-yl)pyrimidine
6-{[3-(hydroxymethyl)-3-propylpiperidin-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1S,5R)-6-(cyclopropylmethyl)-3-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[3,5-difluoro-4-(trifluoromethyl)phenyl]-3-[2-(dimethylamino)ethyl]-3-methylurea
N-benzyl-N-butyl-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-(carbamoylamino)-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
N-{2-[({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]ethyl}acetamide
2-(quinolin-3-yl)-1,3-thiazole-4-carboxamide
1-(4-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-4-oxobutyl)pyrrolidin-2-one
3-{5-chloro-1-methyl-4-[(3-phenoxyazetidin-1-yl)methyl]-1H-pyrazol-3-yl}-5-methyl-1,2-oxazole
[(3R,4R)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-[2-methyl-3-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)-1H-indol-1-yl]acetamide