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1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
4-(4-methoxyphenyl)-3-[1-(pyrrolidin-1-yl)ethyl]-4H-1,2,4-triazole
3-(1,3-benzothiazol-2-yl)-1-[4-(2-phenylpyrimidin-4-yl)piperidin-1-yl]propan-1-one
1-[2-(dimethylamino)ethyl]-5-[4-(pyridin-4-yl)piperidine-1-carbonyl]piperidin-2-one
N-(2-fluoroethyl)-3-{[(2-methyl-1,3-thiazol-4-yl)methyl]sulfamoyl}benzamide
N-[(5-methylthiophen-2-yl)methyl]-2-(2-oxopyrrolidin-1-yl)-N-(pyridin-4-ylmethyl)propanamide
2-{1-[2-(dimethylamino)ethyl]-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl}-N-methyl-N-(2-methylpropyl)acetamide
3-[(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]phenol
1-(propan-2-yl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}piperidine-3-carboxamide
3-methoxy-2-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)benzamide
N-{[3-methyl-7-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-2-sulfonamide
1-(2-methoxyphenyl)-3-(1-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-2-(pyridin-4-ylsulfanyl)acetamide
3-methoxy-2-({3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
[(3-{[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(pyrazin-2-ylmethyl)amine
2-(4-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenyl)-6-(pyridin-2-yl)-3,4-dihydropyrimidin-4-one
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-cyclopropaneamido-N-(2-methoxyethyl)-4-methyl-N-(propan-2-yl)benzamide
2-methoxy-4-({1-[methyl(pyrazin-2-ylmethyl)amino]hex-5-en-2-yl}oxy)pyridine-3-carbonitrile
N-({3-methyl-7-[4-(1H-pyrazol-1-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-sulfonamide
N-(2-chloro-4-fluoro-5-methylphenyl)-4-methanesulfonamidopiperidine-1-carboxamide
N-{1-[1-(2-cyclohexylacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
1-(1-methylpiperidin-4-yl)-N-(propan-2-yl)piperidine-3-carboxamide
N-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-2,3-dihydro-1H-inden-1-amine
4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1λ6-thiomorpholine-1,1-dione
4-{4-[({[(2R,3R,5S)-2-(4-chlorophenyl)-1-ethyl-5-(hydroxymethyl)-5-methylpyrrolidin-3-yl]methyl}amino)methyl]phenyl}but-3-yn-1-ol
8-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
9-(morpholine-4-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[1-(1H-indol-5-yl)ethyl]-1,3-oxazole-4-carboxamide
7-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-amino-6-[4-(2,1,3-benzothiadiazol-4-ylmethyl)piperazin-1-yl]pyrimidin-4-ol
N-[1-ethyl-7-(4-formylpiperazine-1-carbonyl)-2-methyl-1H-1,3-benzodiazol-5-yl]benzenesulfonamide
5-{[1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-5-yl]methyl}-3-propylimidazolidine-2,4-dione
1-(2-{[bis(prop-2-en-1-yl)amino]methyl}phenoxy)-3-[cyclohexyl(methyl)amino]propan-2-ol
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-4-yl)propanamide
1-[2-(dimethylamino)ethyl]-3-{2-[4-(4-fluorophenyl)piperazin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)pyrrolidine-2,5-dione
3-[5-(5-methyl-1,3-oxazol-4-yl)-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
3-{1-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanoyl]piperidin-4-yl}-1,3-oxazolidin-2-one
N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
3,5-dimethyl-1-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidin-3-yl)-1H-pyrazole
3-(2,3-dihydro-1H-inden-2-yl)-5-methyl-5-(1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
2-({2-[1-(4-chlorobenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
4-methyl-N-[2-(pyridin-3-yloxy)phenyl]-1,4-diazepane-1-carboxamide
3-(4-chloro-1H-pyrazol-1-yl)-N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyacetyl)pyrrolidin-3-yl]propanamide
2-{3-[4-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]phenoxy}acetamide
N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]-2-(pyrrolidin-3-yl)benzamide
3-(1-cyclopentyl-1H-pyrazol-5-yl)-1-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-1-methylurea
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{[5-(3,6-dimethylpyrazin-2-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
4-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)morpholine-2-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-(4-phenylbutanoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one