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1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
2-(3-methoxyphenoxy)-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-{4-[(3,4-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}pyridine-4-carboxylic acid
1-(2-methyl-6-propylpyrimidin-4-yl)-N-[2-(propan-2-yloxy)ethyl]piperidin-4-amine
1-(4-chloro-1H-pyrazole-3-carbonyl)-3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine
1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-2-(1H-1,2,3-triazol-1-yl)ethan-1-one
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-[3-(4-fluorophenyl)phenyl]pyrrolidine-2-carboxamide
(3aR,6aS)-2-ethyl-5-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3S,4R)-3-benzyl-4-methyl-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-ol
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(1S,5R)-6-(cyclobutylmethyl)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-cyclopropyl-5-(1,2-oxazol-5-yl)-1-phenyl-1H-1,2,4-triazole
N-[3-(benzylsulfanyl)propyl]pyrrolidine-3-carboxamide
N-(4-fluoro-2-methylphenyl)-3-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)propanamide
4-{1-[(4-ethoxyphenyl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
2-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethan-1-amine
2-{4-[(2,3-dimethoxyphenyl)methyl]-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-(1-benzyl-1H-imidazol-2-yl)-1-(4-methylbenzoyl)piperidine
2-(1-cyclopropanecarbonylpiperidin-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-({1-[6-(4-aminopiperidin-1-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
2-(4-{[5-(3-chlorophenyl)furan-2-yl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
2,5-dimethyl-4-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
N-(1-{7-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
N-butyl-3-methyl-N-(thiophen-3-ylmethyl)furan-2-carboxamide
4-(4-methanesulfonylphenyl)-6-methyl-2-propylpyrimidine
5-{[2-(2-phenylethyl)morpholin-4-yl]methyl}-2,1,3-benzoxadiazole
(2S,4S)-4-amino-N,N-diethyl-1-(1-ethyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)pyrrolidine-2-carboxamide
2-[3-methyl-4-({1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}methyl)-1H-pyrazol-1-yl]ethan-1-ol
N-[(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)methyl]thiophene-2-carboxamide
1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-N-[2-(thiophen-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
(4aS,8aR)-6-(6-aminopyrimidin-4-yl)-1-[2-(cyclohex-1-en-1-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(4-hydroxyphenyl)-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
3-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-4-(1H-pyrazole-4-carbonyl)-1,4-diazepan-2-one
N-{2-[cyclopentyl(methyl)amino]ethyl}-N,6-dimethyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
4-[4-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]phenol
1-methyl-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H-pyrrole-3-carbonitrile
4-(4-fluorophenyl)-N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)benzamide
4-(2,3-dihydro-1H-isoindole-2-carbonyl)-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
N-[(2R,3R)-1'-(3,5-dimethylbenzoyl)-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(3,4-difluorophenyl)methyl]piperidine
(3S,4R)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide
2-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-2,8-diazaspiro[4.5]decane
1-[2-(4-{[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-oxoethyl]pyrrolidin-2-one
3,3-dimethyl-1-({5-[(4-methyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
4-(1-methyl-1H-1,3-benzodiazol-2-yl)phenol
1-methyl-4-[3-(3-phenylpropanoyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one