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1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
ethyl 1-[4-(4-hydroxyphenyl)butan-2-yl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
3-[(3R,4S)-4-(dimethylamino)-1-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]piperidin-3-yl]propanoic acid
4-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-4-yl)pyridine
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-[6-methyl-3-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)quinolin-2-yl]piperidin-3-ol
4-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-2,6-dimethylpyridine
N-{2-[methyl(phenyl)amino]propyl}-1,1-dioxo-1λ6-thiane-4-carboxamide
3-[ethyl({[3-(pyridin-2-ylmethoxy)phenyl]methyl})amino]-1λ6-thiolane-1,1-dione
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]methanol
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl][(2E)-3-(furan-2-yl)prop-2-en-1-yl]methylamine
N-[(7-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-2-(3-fluorophenyl)acetamide
1-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]-3-(1H-pyrazol-4-yl)propan-1-one
1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
4-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidine-1-carbonyl]-1-ethyl-1,2-dihydropyridin-2-one
N-[2-(dimethylamino)-2-(3-methylphenyl)ethyl]-1,3-dimethyl-1H-pyrazole-4-carboxamide
2-[2-(3-fluorophenyl)piperidine-1-carbonyl]-5-methoxy-1H-indole
1-benzyl-N3-cyclopropyl-N5-[(1R)-1-(3-methoxyphenyl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(1S,6R)-3-methyl-N-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
(2,1,3-benzothiadiazol-5-ylmethyl)({[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
3-methanesulfonamido-5-({[(3-methylphenyl)methyl]amino}methyl)-N-phenylbenzamide
7-{2-methylpyrido[2,3-d]pyrimidin-4-yl}-3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-[(2-ethylpyrimidin-5-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
5-acetyl-N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(3aS,6aS)-2-[(3-fluorophenyl)methyl]-5-(thiophen-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
3-[3-(2-ethoxyethoxy)benzoyl]-3,9-diazaspiro[5.5]undecane
1-(2H-1,3-benzodioxol-4-ylmethyl)-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
3-[1-(4-acetylbenzoyl)piperidin-3-yl]-N-[(2-chlorophenyl)methyl]propanamide
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-3-(pyridin-3-yl)propan-1-one
N-{2-[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-4-(1H-pyrazol-1-yl)benzamide
2-methyl-1-{1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]azetidin-3-yl}piperidine
3-{1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}benzoic acid
4-[2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-benzofuran-5-yl]-1-(thiophen-2-ylmethyl)piperidin-4-ol
1-[(2-methoxyphenyl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
1-(cyclohexylmethyl)-3-{[ethyl(methyl)amino]methyl}-3-hydroxypiperidin-2-one
4-(2,3-dihydro-1H-inden-2-yl)-2-[(4-fluorophenyl)methyl]morpholine
(3S)-3-(3-methoxyphenyl)-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
3-[3-(3-chlorophenoxy)azetidin-1-yl]propane-1,2-diol
(4aS,7aR)-N-(4-chlorophenyl)-6,6-dioxo-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
ethyl 1-[(2-ethoxy-2-oxoethyl)carbamoyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
3-ethyl-4-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
1-[2-(dimethylamino)ethyl]-3-(2-fluorophenyl)-3-[2-(4-methyl-3-phenylpiperazin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
1-{3-[(4-methoxyphenyl)amino]piperidine-1-carbonyl}cyclopropane-1-carboxamide
5-fluoro-N2-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N4,N4-dimethylpyrimidine-2,4-diamine
1-(2-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}phenyl)ethan-1-one
(2S,4S)-N-ethyl-4-[2-(5-methyl-1H-pyrazol-1-yl)acetamido]-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide