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N-(2-hydroxy-2-phenylethyl)-N-methyl-1-(4-methylquinazolin-2-yl)piperidine-4-carboxamide
(1R,5R)-3-benzoyl-6-[(3,5-difluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
methyl 3-(3-chlorobenzamido)-6-[(diethylamino)methyl]thieno[2,3-b]pyridine-2-carboxylate
ethyl 1-{1-[2-(benzenesulfonyl)ethyl]-7-oxoazepan-4-yl}piperidine-3-carboxylate
5-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-1-[2-(4-methoxyphenyl)ethyl]piperidin-2-one
(1R,3S)-3-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}cyclopentan-1-amine
[(2S,6S)-4-(quinoline-7-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
5-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)pentan-1-ol
N,5-dimethyl-N-(2-methylpropyl)-4-{[3-(morpholin-4-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
4-[(4-fluorophenyl)methyl]-1-(3-methyl-1H-pyrazole-5-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-ethyl-N-(2-hydroxyethyl)-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
N-{3-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]phenyl}acetamide
2-{[4-(3-methylphenyl)-5-[1-(propan-2-yloxy)ethyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-(dimethylamino)-N,4-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyrimidine-5-carboxamide
1-(4-amino-5-methylpyrimidin-2-yl)-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
[(1R,5S,6R)-3-azabicyclo[3.1.0]hexan-6-ylmethyl](2-methoxyethyl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
1-(3-methylfuran-2-carbonyl)-N-(6-methylpyridin-3-yl)piperazine-2-carboxamide
4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N,N-dimethyl-1-[4-(1,3-oxazol-5-yl)benzenesulfonyl]azepan-4-amine
1,9-dimethyl-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-[3-(thiophen-2-yl)-1H-pyrazol-1-yl]acetamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]acetamide
N-[3-(4-chlorophenoxy)propyl]-N-methyl-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N2-[2-(dimethylamino)ethyl]-N5-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2,5-dicarboxamide
1-[(2-fluorophenyl)methyl]-N-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-amine
5-(2,5-dimethylphenoxymethyl)-N-[(5-methylpyrazin-2-yl)methyl]-1,2-oxazole-3-carboxamide
(2S)-2-{4-phenyl-5-[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]-1H-imidazol-1-yl}propanamide
6-methoxy-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-(2-chloro-5-fluorophenyl)-4-(prop-2-en-1-yl)piperazine-1-carboxamide
(3aR,6aR)-2-cyclopentyl-5-[(1-methyl-1H-indol-6-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(1R,3R)-3-aminocyclopentyl]-5-chloro-1,3-dimethyl-1H-pyrazole-4-sulfonamide
methyl 3-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-methyl-5-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrazine
3-[1-(1-hexylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-1-ol
3-{[3-(2-phenylacetyl)piperidin-1-yl]methyl}-1,2-dihydroquinoxalin-2-one
methyl[(1-methylpyrrolidin-2-yl)methyl]({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)amine
3-[2-(2-chloro-4-fluorophenyl)acetyl]-9-methoxy-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylacetamide
2-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]-N-(2-fluoro-4-methylphenyl)acetamide
1-[(6-fluoroquinolin-2-yl)methyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(3R,4R)-4-amino-1-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}piperidin-3-ol
N-cyclopropyl-N-[(3-ethoxyphenyl)methyl]-2-(2,2,3,3-tetrafluoropropoxy)acetamide
{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
N-[2-(azepan-1-yl)ethyl]-5-chloro-N-ethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[3-(naphthalene-2-carbonyl)piperidin-1-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
1-{2-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]piperidin-1-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
N-[3-(2-ethylphenoxy)propyl]-N-methyl-1,1-dioxo-1λ6-thiane-4-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
N-(2-{7-[(5-ethylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-(4-fluorophenyl)acetamide
1-[1-(1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)piperidin-3-yl]ethan-1-one