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(2S)-N-(1-methyl-4-phenyl-1H-pyrazol-5-yl)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
5-{[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]methyl}-1-phenyl-1H-1,2,3,4-tetrazole
1,3-dimethyl-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
6-methyl-2-[(2-methylphenyl)methyl]-N-(1,2-oxazol-3-ylmethyl)-4-oxo-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-(2-chloro-6-methylphenyl)-3-(naphthalene-2-carbonyl)piperidine-1-carboxamide
5-methyl-1-(4-methylphenyl)-4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperazin-2-one
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
7-fluoro-3-[({[1-(morpholin-4-yl)cyclohexyl]methyl}amino)methyl]-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one
1-(2-methoxyphenyl)-4-{1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-3-yl}piperazine
1-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-yl]-2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)ethan-1-one
methyl 7-oxo-3-(5-propyl-1,2-oxazole-3-carbonyl)-9-[3-(pyridin-4-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{4-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-pyrazol-5-yl}-1H-1,2,3,4-tetrazole
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-(1-propylpiperidin-4-yl)acetamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl](2-methoxyethyl)amine
(2S,4R)-1-[(4-chlorophenyl)methyl]-4-{[(9-ethyl-9H-carbazol-3-yl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
6-methyl-2-[({4-methyl-6H,7H,8H-cyclopenta[g]quinolin-2-yl}amino)methyl]-3,4-dihydropyrimidin-4-one
N-[cyclopropyl(4-methoxyphenyl)methyl]-3-(pyridin-4-yl)propanamide
9-(2,4-difluorobenzoyl)-6-(4-methoxyphenyl)-6,9-diazaspiro[4.5]decan-7-one
2,5-dimethyl-N-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidine
N-({1-[(3-chloropyridin-4-yl)methyl]pyrrolidin-3-yl}methyl)-2-hydroxybenzamide
N-{5H,6H,7H,8H,9H,10H-cyclohepta[b]indol-2-ylmethyl}-4-(1H-1,2,3,4-tetrazol-1-yl)butanamide
N-(2H-1,3-benzodioxol-5-yl)-6-[2-(cyclohex-1-en-1-yl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
N-methyl-2-(pyridin-4-yl)-N-(thian-4-yl)quinoline-4-carboxamide
N-[4-(2-fluorophenoxy)phenyl]-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine-2-carboxamide
N-cyclopentyl-1-[(4-methoxyphenyl)methyl]-5-[3-(pyridin-2-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-(3-methylcinnolin-5-yl)piperidine-1-carboxamide
3-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(naphthalen-1-yl)urea
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2-oxo-2-(pyridin-3-yl)acetamide
(2R)-3-methyl-2-[2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamido]butanamide
1-(4-acetylpiperazin-1-yl)-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propan-1-one
4-[(2-fluorophenyl)methyl]-3-(pyrazin-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4S)-4-amino-1-(6-aminopyridine-3-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
N-(furan-2-ylmethyl)-2-oxo-N-(pyridin-2-ylmethyl)-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
1-[1-(azepan-1-yl)-2-methylpropan-2-yl]-3-(1-propyl-1H-1,2,4-triazol-3-yl)urea
(3S,9aR)-8-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(1H-indol-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[4-(4-{[(5-chloro-2-fluorophenyl)formamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-5-(methoxymethyl)furan-2-carboxamide
2-[2-(dimethylamino)ethyl]-8-{2-[methyl(phenyl)amino]acetyl}-2,8-diazaspiro[5.5]undecan-3-one
6-methoxy-3-methyl-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}-1-benzofuran-2-carboxamide
2-(3-{3-[5-(trifluoromethyl)pyridin-2-yl]phenyl}-1H-pyrazol-1-yl)ethan-1-ol
6-(2,5-dimethylfuran-3-yl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
dimethyl(2-{2-[1-(quinoline-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
3-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
(3S)-1-[4-(1H-pyrazol-5-yl)benzoyl]piperidin-3-amine
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
N-(pyridin-3-ylmethyl)-3-{[1-(thiophen-3-ylmethyl)piperidin-4-yl]oxy}benzamide
1-(adamantan-1-yl)-4-[(5-chlorofuran-2-yl)methyl]piperazine
5-[1-(4-methyl-1H-imidazole-2-carbonyl)pyrrolidin-2-yl]-N-(pyridin-3-yl)thiophene-2-carboxamide
ethyl 1-{[2-(methylsulfanyl)phenyl]carbamoyl}-4-(oxan-2-ylmethyl)piperidine-4-carboxylate