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N-(1,3-dimethyl-1H-pyrazol-5-yl)-3-{[ethyl(pyridin-4-ylmethyl)amino]methyl}benzamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-(propan-2-yl)benzamide
N-[2-(4-methoxyphenyl)phenyl]-1-(1H-pyrazole-4-carbonyl)pyrrolidine-2-carboxamide
(3aS,6aS)-2-[(4-cyanophenyl)methyl]-5-[3-(methylsulfanyl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-1,2-oxazinane
7-(cyclohexylmethyl)-2-(thian-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
3-{1-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(1,2-oxazolidin-2-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
1-{[4-(2-methylpropyl)phenyl]methyl}-4-(prop-2-en-1-yl)-1,4-diazepan-5-one
7-[1-(4-chlorophenyl)cyclobutanecarbonyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-(2,4-dimethoxyphenyl)-6-(1H-pyrazol-1-yl)pyrimidine
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-4-yl}propanamide
N-(4-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]acetamido}-2-methoxyphenyl)-3-methylbutanamide
2-amino-8-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
(3aS,6aS)-2-(dimethylcarbamoyl)-5-(4-phenoxybutyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(5-chloro-2-methoxyphenyl)-2-[4-(2-methoxyethyl)piperazin-1-yl]acetic acid
2-[(4-methoxyphenyl)methyl]-N-[2-(morpholin-4-yl)ethyl]-1,3-benzoxazole-6-carboxamide
2-(2-{1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
5,7-dimethyl-N-[(1-methylpiperidin-2-yl)methyl]pyrido[2,3-d]pyrimidin-4-amine
methyl (2S,4S)-1-methyl-4-{2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamido}pyrrolidine-2-carboxylate
3-methyl-5-{2-oxo-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
8-(benzenesulfonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[(5,8-dimethoxy-4-methylquinolin-2-yl)amino]propan-1-ol
1-(diphenylmethyl)-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)urea
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-(2-methoxyethoxy)ethan-1-one
2-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazole
N,N-dimethyl-6-(3-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidin-4-amine
2-(3-phenylpropyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1,3-benzoxazole-5-carboxamide
1-(1-benzylpiperidin-4-yl)-N-(2-methoxyethyl)-N-methylpiperidine-3-carboxamide
1-[(3aS,6aS)-5-(4-cyclopentylpyrimidin-2-yl)-octahydropyrrolo[3,4-b]pyrrol-1-yl]-3-(methylsulfanyl)propan-1-one
4-[2-hydroxy-3-(2-methylphenoxy)propanoyl]-1-[(3-methylphenyl)methyl]piperazin-2-one
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[(2-methoxypyridin-3-yl)methyl]piperidine-4-carboxylic acid
(1R,9S)-5-amino-3-(1-phenyl-1H-pyrazol-4-yl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-[(2-fluorophenyl)methyl]-1,4-diazepane
3-(3-methylbutyl)-8-(1-methylcyclopropanecarbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-chloro-N-(2-methoxyethyl)-4-[(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)oxy]benzamide
10-[4-(4-fluorophenyl)piperazine-1-carbonyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
methyl 4-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butanoate
3-benzyl-4-[5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperazin-2-one
N-cyclopropyl-5-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-[(3R,4S)-1-(2,6-difluoro-3-methylbenzoyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-(propan-2-yl)-1,3-thiazole-2-carboxamide
2-[5-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-methyl-N-[(5-methylfuran-2-yl)methyl]benzamide
(4aS,7aR)-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-(1-benzothiophen-3-yl)-N-(1,4-dioxan-2-ylmethyl)-N-methyl-3-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]pyridin-2-amine
5-(4-acetyl-2-methoxyphenoxymethyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]-1,2-oxazole-3-carboxamide
1-{5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidine-3-carboxamide
8-(2-ethoxyacetyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one