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1-(4-{4-[3-(dimethylamino)pyrrolidine-1-carbonyl]phenoxy}piperidin-1-yl)-2-methoxyethan-1-one
(2S,4R)-4-amino-1-(2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
1-(1-benzoylpiperidin-3-yl)-4-(2-methoxyphenyl)piperazine
3-(4-methoxy-3,5-dimethylbenzoyl)-1-phenylmethanesulfonylpiperidine
N-[2-(1H-indol-3-yl)ethyl]-6-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[(3R,4S)-1-[(4,6-dimethylpyrimidin-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
N-cyclopentyl-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
4-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one
methyl 3-(furan-2-amido)-1-(2-methoxyethyl)-5-{[(3-methoxyphenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[1-(3-methylbut-2-enoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
2-(3,4-dichlorophenyl)-N-(dimethyl-1,2-oxazol-4-yl)morpholine-4-carboxamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N3-benzyl-N3-butyl-N5-(2-methoxyethyl)-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(acetamidomethyl)-N-(2-propylphenyl)-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
(4aS,8aR)-2-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-decahydroisoquinoline
6-[4-(2-chlorophenoxy)piperidine-1-carbonyl]-1,3-benzothiazole
9-methoxy-4-[(4-methyl-1H-imidazol-5-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-1-methyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
2-{4-[(3,4-difluorophenyl)methyl]-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-(carbamoylmethyl)-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}piperidine-4-carboxamide
N-[(2-aminopyrimidin-5-yl)methyl]-N-methyl-4-(1H-pyrazol-3-yl)benzamide
5-acetamido-N-[2-(2-fluorophenyl)ethyl]-1-(2-methoxyethyl)-2-(pyridin-2-yl)-1H-1,3-benzodiazole-7-carboxamide
3-[cyclopentyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amino]propane-1,2-diol
1-(3,5-dimethylphenyl)-4-(oxolan-3-ylmethyl)piperazin-2-one
2-{[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]methyl}quinolin-4-ol
1-(2-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
1-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-imidazole
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2H-1,3-benzodioxole-5-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-(pyrrolidin-1-yl)benzamide
methyl 3-[(3S,4R)-1-[(2-hydroxy-5-methoxyphenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoate
N-[(3R,4R)-1-[3-(3-chlorophenyl)propanoyl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
N-methyl-1-[2-(piperazin-1-yl)ethyl]-N-(quinolin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[4-(4-fluoro-3-methoxyphenyl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]pyridine-3-carboxamide
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N,1,3-trimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-(4-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
methyl 1-(2-methoxyethyl)-3-(2-phenylacetamido)-5-[(4,4,4-trifluorobutan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1R,9aR)-1-{[4-(4-methylpyridin-2-yl)piperazin-1-yl]methyl}-octahydro-1H-quinolizin-1-ol
3-[(dimethylcarbamoyl)methyl]-2-oxo-1-(2-phenylethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
N-cyclohexyl-3-(2,5-dioxoimidazolidin-4-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]propanamide
6-chloro-N-[(1-ethylpyrrolidin-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-5-sulfonamide
3-chloro-N-cyclopentyl-4-{[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]oxy}benzamide
(5-{1-[(4-methyl-1,3-benzoxazol-2-yl)methyl]-4-phenyl-1H-imidazol-5-yl}furan-2-yl)methanol
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-6-hydroxy-1,4-oxazepane-4-carboxamide
14-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-[(1S,2R)-2-aminocyclobutyl]-3-(2-oxo-1,2-dihydropyridin-1-yl)propanamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-3-(3-methoxyphenyl)-1H-pyrazole
5-methoxy-3-methyl-2-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]-1H-indole
{2-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]-1,3-thiazol-4-yl}methanol
4-(2-methylpropyl)-1-(thiophene-2-carbonyl)-1,4-diazepan-5-one