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(1S,4S)-5-[(2S)-2-amino-4-hydroxybutanoyl]-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
4,6-dimethyl-2-oxo-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,2-dihydropyridine-3-carboxamide
N-(3-fluorophenyl)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
1-methyl-4-(4-methylpyridine-3-carbonyl)piperazine-2-carboxylic acid
N6-benzyl-N5-[(1-methyl-1H-imidazol-2-yl)methyl]-N5-(propan-2-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-(2-methoxy-2-phenylacetyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4,4,4-trifluoro-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]butan-1-one
N-ethyl-3-(3-methoxyphenyl)-N-(pyridin-4-ylmethyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
1-butyl-3-cyclopropyl-5-{6-methylpyrazolo[1,5-a]pyrimidin-3-yl}-1H-1,2,4-triazole
3-[1-(3-cyanophenyl)-N-methylformamido]-N-methylpropanamide
N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-4-(pyridin-4-yl)pyrimidin-2-amine
2-(1,6-dimethyl-1H-indole-2-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-3,6-dimethyl-1-benzofuran-2-carboxamide
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-[3-(5-methylfuran-2-yl)-1H-pyrazol-1-yl]acetamide
4-[(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-2-yl)methyl]morpholine
5-(dimethylamino)-2-[(3-methylquinoxalin-2-yl)methyl]-2,3-dihydropyridazin-3-one
4-(hydroxymethyl)-1-{6-methyl-2H-[1,3]dioxolo[4,5-g]quinolin-8-yl}piperidin-4-ol
N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
N,1-dimethyl-6-oxo-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]-1,4,5,6-tetrahydropyridazine-3-carboxamide
1-{2-[(3S)-3-(dimethylamino)azepan-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
3-({1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-yl}amino)piperidin-2-one
4-(4-ethoxy-3-methylphenyl)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-4-oxobutanamide
1-[1-(methoxymethyl)cyclopropanecarbonyl]-2-(thiophen-2-yl)azetidine
3-{5-[2-(2H-indazol-2-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
2-[methyl(pyridin-3-ylmethyl)amino]-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]acetamide
1-cyclohexyl-3-(cyclopropylmethyl)-5-(4-hydroxypiperidine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(oxolan-2-ylmethyl)amine
3-[1-(2-methoxypyridin-3-yl)-1H-imidazol-2-yl]-6,8-dimethyl-1,2-dihydroquinolin-2-one
N-({3-[(2-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)-N-(pyridin-4-ylmethyl)propanamide
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3,4-dimethylphenyl)urea
N-(4-{1-[1-(3-methylpyridin-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}phenyl)acetamide
4-(2,6-difluorobenzenesulfonyl)-9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}pyrrolidin-3-ol
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine-4-carboxamide
1-(7-methoxy-4-methylquinazolin-2-yl)-N-[1-(thiophen-3-yl)propan-2-yl]piperidin-4-amine
4-{3-[(2-phenylethyl)carbamoyl]piperidin-1-yl}-N-(propan-2-yl)piperidine-1-carboxamide
(4aS,8aR)-2-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-decahydroisoquinoline
methyl 3-benzamido-5-[(2,1,3-benzothiadiazol-5-ylmethyl)amino]-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[3-(morpholin-4-yl)piperidin-1-yl]-3-(pyridin-2-yl)propan-1-one
2-({6-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
methyl 3-[5-(4-acetamidophenyl)-4-phenyl-1H-imidazol-1-yl]propanoate
1-(3-oxo-3-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(1-oxo-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}butan-2-yl)-2,3-dihydro-1H-isoindol-1-one
2-cyclobutanecarbonyl-7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-6-one
3-(3-ethyl-1,2,4-oxadiazol-5-yl)-2-methyl-N-(pyridin-3-ylmethyl)aniline
3-(3-methoxybenzoyl)-1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine
1-(furan-3-ylmethyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
N-[2-(dimethylamino)ethyl]-5-(quinolin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(1S,4S)-2-[5-(3-fluorophenyl)-1,2,4-triazin-3-yl]-2-azabicyclo[2.2.1]heptane
2-methyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}furan-3-carboxamide