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3-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
[(2S,4R,5R)-5-(2-fluorophenyl)-1-methyl-4-[({[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amino)methyl]pyrrolidin-2-yl]methanol
2-methoxy-N-({5-[(3,4,5-trifluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
1-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
4-[(2-fluorophenyl)methyl]-1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
1-methyl-9-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
5-(oxane-4-carbonyl)-3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-methyl-2-oxo-N-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
1-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-methylbutan-1-one
3-(3-hydroxy-3-methylbutyl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}benzamide
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-[3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]-2-(pyridin-4-yl)ethan-1-one
1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N,N-dimethyl-5-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-[2-(methylsulfanyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
propyl 3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
2-(dimethylamino)-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-(3-methylphenyl)acetamide
5-butyl-1-(2-methoxyphenyl)-4-(1-methyl-1H-pyrazole-4-carbonyl)piperazin-2-one
9-hydroxy-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
3-ethyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-4-yl}urea
(3-{2-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}propyl)dimethylamine
1-benzyl-3-(2-methylphenyl)-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
6-{2-[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}-1H-indazole
2-amino-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1,3-benzothiazole-5-carboxamide
1-(1-acetylpiperidine-2-carbonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
[(3S,5R)-1-(5-methoxypyrimidin-2-yl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
1-[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]-4-phenylpiperazine
(1S,5R)-6-benzyl-3-{2-methylthieno[2,3-d]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-propoxyethyl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-{4-[({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]thiophen-2-yl}ethan-1-one
4-[4-phenyl-5-(2-phenylethyl)-1H-imidazol-2-yl]pyrrolidin-2-one
2-benzyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1,3-thiazole-4-carboxamide
2-methoxy-N-[(1R,2S)-2-phenylcyclopropyl]pyrimidine-5-carboxamide
methyl({[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl})[1-(1,2-oxazol-3-yl)ethyl]amine
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-5-acetylthiophene-3-carboxamide
1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-2-[2-(thiophen-2-yl)ethyl]piperidine
1-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(2-methoxybutanoyl)-2,8-diazaspiro[4.5]decan-3-one
1-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
6-(3-methyl-3-phenylpiperidine-1-carbonyl)-1,2,3,4-tetrahydroquinoxaline-2,3-dione
(5S,9aS,9bS)-2-phenyl-5-(quinolin-5-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(oxan-4-ylmethyl)amine
(2S)-1-acetyl-N,N-bis(furan-2-ylmethyl)pyrrolidine-2-carboxamide
2-{[4-(3-hydroxy-3-methylbutyl)phenyl]formamido}-N-(propan-2-yl)acetamide
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(1,3-thiazol-4-ylmethyl)piperidine
1-(5-phenyl-1,2,4-oxadiazol-3-yl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
{3-[(2-fluorophenyl)methyl]-1-(pyrimidin-2-yl)piperidin-3-yl}methanol
2-[1-(2,2-dimethylpropyl)-4-{[3-(methylsulfanyl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
3-methyl-8-{[4-(2-methylphenyl)phenyl]methyl}-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione