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N-cyclopropyl-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-[(3-methylthiophen-2-yl)methyl]benzamide
{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
1-[7-(1-benzothiophen-3-yl)-9-[2-(pyridin-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
4-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)-N-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}benzamide
1-({1-[2-(hydroxymethyl)pyridin-4-yl]piperidin-3-yl}methyl)pyrrolidin-2-one
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
3-(1-{[5-(oxan-2-yl)thiophen-2-yl]methyl}piperidin-4-yl)-N-(pyridin-3-ylmethyl)propanamide
(3R)-1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}pyrrolidin-3-ol
(3aS,6aS)-2-cyclobutanecarbonyl-5-(pyrimidin-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}acetamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(2-methoxynaphthalen-1-yl)methyl]piperazin-2-yl}ethan-1-ol
4-ethyl-1-methyl-3-(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[(dimethylamino)methyl]-N-[1-(pyrrolidin-1-ylmethyl)cyclohexyl]benzamide
N,1,3-trimethyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(4aS,7aR)-1-benzoyl-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
2-(furan-3-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
1-methyl-5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazole
2-(5-{[3-(hydroxymethyl)-4-methylpiperazin-1-yl]methyl}furan-2-yl)benzonitrile
(1,4-dioxan-2-ylmethyl)({[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl})methylamine
3-({1-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]pyrrolidin-3-yl}methyl)benzoic acid
benzyl({[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
N-[(3,4-difluorophenyl)methyl]-3-{1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidin-3-yl}propanamide
[4-({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)-1,4-oxazepan-6-yl]methanol
4-[2-(4-chloro-1H-pyrazol-1-yl)acetyl]-1-(4-methylphenyl)piperazin-2-one
4-hydroxy-N-methyl-2-(phenoxymethyl)-N-[1-(pyridin-3-yl)propyl]pyrimidine-5-carboxamide
ethyl 4-{[3-(morpholin-4-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
methyl 6-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-1-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]propan-1-one
4,6-dimethyl-2-oxo-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
6-{2-[1-(2-methylpropyl)piperidin-2-yl]ethyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-({[(3-fluorophenyl)methyl]amino}methyl)-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
ethyl 4-(oxan-2-ylmethyl)-1-(quinolin-6-ylmethyl)piperidine-4-carboxylate
methyl 1-{2-[(1-acetylpiperidin-4-yl)oxy]-5-chlorobenzoyl}piperidine-2-carboxylate
N-(2-phenylethyl)-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{3-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidin-1-yl}-2-(pyridin-2-yl)ethan-1-one
(2S,4S)-1-[(2-aminopyridin-3-yl)methyl]-4-benzamido-N-ethylpyrrolidine-2-carboxamide
N-[3-(3-oxopiperazin-1-yl)propyl]-4-propylpyrimidine-5-carboxamide
5-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-4-methyl-2-(propan-2-yl)pyrimidine
3-[3-(3,4-dimethoxybenzoyl)piperidine-1-carbonyl]-1H-indazole
1-{2-[1-(2-fluoro-4-methylbenzenesulfonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
1-[3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)propyl]pyrrolidin-2-one
1-methyl-4-(1-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-4-phenyl-1H-imidazol-5-yl)piperidine
5-methyl-4-[4-(pyrrolidin-3-yl)piperazin-1-yl]pyrimidin-2-amine
1-[(3-acetylphenyl)methyl]-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
1-{2-oxo-2-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethyl}azepan-2-one
2-{1-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
3-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-7-methyl-3H,4H-thieno[3,2-d]pyrimidin-4-one
1-(4-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-6-hydroxy-1,4-diazepan-1-yl)ethan-1-one