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N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-1-methylcyclopropane-1-carboxamide
N-[2-(1H-imidazol-1-yl)ethyl]-2-(morpholin-4-yl)-6-phenylpyridine-3-carboxamide
N,2,6-trimethyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]pyrimidine-4-carboxamide
3-(azocan-1-yl)-N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]propanamide
N-[1-(2-chlorophenyl)cyclopropyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1-(oxan-3-ylmethyl)-1H-imidazole
N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
ethyl 4-[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]piperidine-1-carboxylate
1-{1-[4-(3-fluorophenyl)benzoyl]piperidin-4-yl}-2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazole
2-(4-methoxyphenoxymethyl)-4-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,3-oxazole
2-[(3-methoxyphenyl)methyl]-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[4.5]decan-3-one
2-[(adamantan-1-yl)amino]-N-[1-(4-methylphenyl)ethyl]acetamide
1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(2-phenylethyl)piperidine-4-carboxamide
N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H,4H,6H,7H-pyrano[4,3-c]pyrazole-3-carboxamide
1,3-dimethyl-N-[2-(4-{[methyl(naphthalen-1-ylmethyl)amino]methyl}phenoxy)ethyl]-1H-pyrazole-5-carboxamide
1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
3-(4-hydroxyphenyl)-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-5-carboxamide
N-cyclohexyl-3-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propanamide
(4aR,8aS)-1-[2-(diethylamino)ethyl]-6-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-decahydro-1,6-naphthyridin-2-one
3-{[(butan-2-yl)(thiophen-3-ylmethyl)amino]methyl}-7-fluoro-1,2-dihydroquinolin-2-one
4-(4-{2,5-dioxo-4-propyl-1-[2-(thiophen-2-yl)ethyl]imidazolidin-4-yl}piperidin-1-yl)-N,N-dimethyl-4-oxobutanamide
1-(cyclohexylmethyl)-3-hydroxy-3-({[(1r,4r)-4-hydroxycyclohexyl]amino}methyl)piperidin-2-one
1-[(4aR,8aR)-6-[2-(4-fluorophenyl)acetyl]-decahydro-1,6-naphthyridin-1-yl]-2-(4-methylphenoxy)ethan-1-one
3-{2-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
9-(cyclopropylmethyl)-4-(furan-3-ylmethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-(2,6-dimethoxyphenyl)-2-ethyl-1,3-benzoxazole
N-methyl-N-(2-phenyl-1-{1-[(2E)-3-phenylprop-2-enoyl]piperidin-4-yl}ethyl)thiophene-3-carboxamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)isoquinoline-3-carboxamide
2-[1-(2-hydroxyethyl)-5-[({6-methylthieno[2,3-d]pyrimidin-4-yl}sulfanyl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
3-[(3R,4S)-1-(7-methyl-1-benzofuran-2-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
N-cyclopentyl-1-[(4-methoxyphenyl)methyl]-5-[(5-methylfuran-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-pyrazole-3-carboxamide
(3R,4R)-1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
3-ethyl-5-methyl-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-1,2-oxazole-4-carboxamide
5-cyclopropanecarbonyl-1'-(2-methylpyrimidine-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{[4-(oxolan-3-ylmethoxy)phenyl]methyl}-4-(1H-pyrazol-1-yl)-N-(pyridin-3-ylmethyl)benzamide
N-[(2R,3R)-2-methoxy-1'-(4-methylpentanoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
5-methyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-1-propyl-1H-pyrazole-4-carboxamide
N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
2-chloro-4-fluoro-N-[1-(3-phenylpropyl)piperidin-3-yl]benzamide
(1r,4r)-4-{[2-(dimethylamino)-2-(3-methylphenyl)acetamido]methyl}cyclohexane-1-carboxamide
N-[2-(pyridin-2-yl)ethyl]-6-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(4-methoxyphenyl)-1-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]ethan-1-one
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
4-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
5-{1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
7-(2-aminophenyl)-2,3-dihydro-1,4-benzodioxine-6-carboxylic acid
1-[2-(ethoxymethyl)-7-(furan-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-2,5-dihydro-1H-pyrrole
N-{[7-(3-fluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}propane-1-sulfonamide