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[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)methylamine
4-[({[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-1-ethylpyrrolidin-2-one
4-benzyl-1-[1-(methylsulfanyl)propan-2-yl]piperidine
2-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}-2-(5-fluoro-2-methoxyphenyl)acetic acid
N-(furan-3-ylmethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N'-cycloheptyl-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}butanediamide
1-(2-chlorophenyl)-3-{1-[1-(3-hydroxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-[(4-methylphenyl)methyl]-1,3-oxazole-4-carboxamide
N-(2-methylpropyl)-2-(4-oxo-1,4-dihydropyridin-1-yl)-N-(propan-2-yl)acetamide
N-ethyl-N-[2-(4-fluorophenoxy)ethyl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
4-{1-[(5-ethylfuran-2-yl)methyl]piperidin-3-yl}-5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidine
2-(dimethyl-1,2-oxazol-4-yl)-N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
3-[3-(2-methoxyethoxy)phenyl]-1-[1-(pyridin-4-yl)propyl]urea
N-methyl-N-{1-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]-2-phenylethyl}thiophene-3-carboxamide
1-(1-ethyl-1H-pyrazole-3-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
(4aR,8aS)-6-[(3,5-dimethoxyphenyl)methyl]-1-[2-(3-fluorophenyl)ethyl]-decahydro-1,6-naphthyridin-2-one
3-{5-[3-(methylsulfanyl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-(morpholin-4-yl)propan-1-one
4,5-dimethyl-3-[2-(2-methyl-2,3-dihydro-1H-indol-1-yl)-2-oxoethyl]-2,3-dihydro-1,3-oxazol-2-one
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{[4-(3-chloro-4-fluorophenyl)-1H-1,2,3-triazol-1-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
8-[(3-hydroxyphenyl)methyl]-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)piperazin-2-one
1-{4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
2-methyl-5-(2-{2-[(1-methylpiperidin-4-yl)amino]ethyl}morpholin-4-yl)-2,3-dihydropyridazin-3-one
8-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(2-hydroxyethyl)-N-methyl-1-[1-(3-phenylpropyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
2-cyclopentyl-9-(6-methyl-2-propylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]({1-[(2-fluorophenyl)methyl]-2-methyl-1H-indol-3-yl}methyl)amine
1-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-N,N-dimethylpyrrolidin-3-amine
N-(2-methoxyethyl)-1-{1-[2-(pyridin-3-yl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
3-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]benzoic acid
3-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(3,5-difluorophenyl)methyl]-8-{2-[ethyl(methyl)amino]acetyl}-2,8-diazaspiro[4.5]decan-3-one
1-methyl-3-(4,4,4-trifluorobutyl)-1H,2H,3H-imidazo[4,5-c]pyridin-2-one
4-[1-(3,5-dimethyl-1-benzofuran-2-carbonyl)piperidin-4-yl]thiomorpholine
2-(3,3-dimethylbutyl)-6,7-dimethoxyquinazolin-4-amine
N-[2-fluoro-5-({[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]carbamoyl}amino)phenyl]-2-methylpropanamide
3-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}-N-methylpyridin-2-amine
2-{1,4-bis[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
methyl 4-({3-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)benzoate
5-(2,6-difluorophenoxymethyl)-N-(1H-imidazol-2-ylmethyl)-N-methyl-1,2-oxazole-3-carboxamide
N-[1-(4-chlorophenyl)cyclobutyl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
4-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine-1-sulfonamide
7-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-[2-(azepan-1-yl)-2-phenylethyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
7-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-[1-(2-cyclopentylacetyl)piperidin-4-yl]-N-[2-(dimethylamino)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-cyclopropyl-N-(2,3-dihydro-1H-inden-2-yl)-1H-pyrazole-5-carboxamide
1-[(2-chloro-4,5-dimethoxyphenyl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one