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{5-[1-(2H-1,3-benzodioxol-5-ylmethyl)-4-phenyl-1H-imidazol-5-yl]furan-2-yl}methanol
6-[(3-fluorophenyl)methoxy]-1-(2-phenylethyl)-4-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-1,4-diazepan-2-one
N-[1-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)pyrrolidin-3-yl]acetamide
3-{5-[2-(3-chloro-4-hydroxyphenyl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
(2-methylpropyl)({[4-(1H-pyrazol-1-yl)phenyl]methyl})(pyridin-2-ylmethyl)amine
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-phenylacetamide
2-{2-[5-(methoxymethyl)thiophene-2-carbonyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
(4aS,7aR)-1-(1-methyl-1H-pyrazole-4-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
1-ethyl-4-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]piperazine-2,3-dione
N3-[2-(cyclohex-1-en-1-yl)ethyl]-1-[(2-methoxyphenyl)methyl]-N5-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(2S,4R)-4-(dimethylamino)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylic acid
(1S,5R)-6-(cyclopropylmethyl)-3-[3-(4-methylphenyl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2,3-dimethyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}quinoxaline-6-carboxamide
N-(3-chloro-4-fluorophenyl)-3-{1-[(2,2-dimethyloxan-4-yl)methyl]piperidin-4-yl}propanamide
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-{[1-(dimethylamino)cyclohexyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2,3-difluoro-4-methoxy-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]benzamide
7-[(2-chlorophenyl)methyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-[1-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)piperidin-4-yl]pyrazolo[1,5-a]pyridine-7-carboxamide
5-(4-methylbenzoyl)-3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}oxolane-2-carboxamide
methyl 3-(cyclobutylmethoxy)-5-[3-(hydroxymethyl)morpholine-4-carbonyl]benzoate
2-[2-(4-fluorophenyl)azetidine-1-carbonyl]-5-methoxy-1-methyl-1H-indole
2-{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}-1,2-oxazinane
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
2-[(6-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}pyrimidin-4-yl)amino]ethan-1-ol
2-cyclopentyl-9-[(5-fluoro-2-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
1-({1-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]piperidin-4-yl}methyl)pyrrolidin-2-one
5-{2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-(4-fluorophenyl)-2-{[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethan-1-ol
1-[(3,4-difluorophenyl)methyl]-3-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
N-[(2-chlorophenyl)methyl]-3-[1-(5-methyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]propanamide
({4-cyclopropyl-5-[1-(4-methylpyrimidine-5-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-[(5-methylfuran-2-yl)methyl]-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
N,N-dimethyl-2-{3-oxo-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-8-yl}acetamide
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-5-cyclopropyl-1,3,4-oxadiazol-2-amine
3-(2-methoxyethyl)-1-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxylic acid
[4-methyl-5-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-4H-1,2,4-triazol-3-yl]methanol
2-(3-hydroxypropyl)-8-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-2-(1-methyl-1H-pyrrol-3-yl)acetamide
1-(cyclohexylmethyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-{[2-(3-chlorophenyl)-7-methylquinolin-3-yl]methyl}-N-(3-methoxypropyl)oxolane-2-carboxamide
1-(dimethyl-1,2-oxazole-4-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
(1R,5S,6S)-N,N-bis(pyridin-3-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
3-{2-[4-(4-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}-3-(4-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
N-({7-[3-(5-methylfuran-2-yl)butyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-2-carboxamide
5-ethyl-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1,3-oxazole-4-carboxamide
pyridin-2-yl(4-{[4-(pyrrolidin-1-yl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol