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1-{2-[(4-methoxy-4-methylpentan-2-yl)amino]ethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
2-(dimethylamino)-2-(3-fluorophenyl)-N-(4-hydroxybutyl)acetamide
3-chloro-N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-6-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide
3-[(oxolan-3-yl)sulfamoyl]-N-[2-(1,3-thiazol-4-yl)ethyl]benzamide
N-(isoquinolin-5-yl)-3-(2-methylpiperidin-1-yl)azetidine-1-carboxamide
N-methyl-N-(oxan-4-ylmethyl)-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
1-cyclopentanecarbonyl-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-4-carboxamide
(1-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)(thiophen-2-yl)methanol
2-(4-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]pyrrolidin-3-yl}piperidin-1-yl)pyrimidine
N,N-dimethyl-2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)-2-phenylacetamide
N-(adamantan-1-ylmethyl)-N,1-dimethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
({4-[2-(1-cyclohexanecarbonylpiperidin-2-yl)ethoxy]phenyl}methyl)(methyl)(thiophen-2-ylmethyl)amine
N-{1-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
1-[1-(2-cyclopropylpyrimidine-5-carbonyl)piperidin-4-yl]piperidin-3-ol
N-(furan-2-ylmethyl)-1-(2-methylpropyl)-4-oxo-5-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-1,4-dihydropyridine-3-carboxamide
4-({4-[(2-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
N-[2-(adamantan-1-yl)ethyl]-1-ethyl-N-methyl-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(pyridin-4-yl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]quinoline-4-carboxamide
1-(morpholin-4-yl)-2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}ethan-1-one
7-{[2-(trifluoromethoxy)phenyl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
3-(2,5-dihydro-1H-pyrrole-1-carbonyl)-N-[(3-methylthiophen-2-yl)methyl]aniline
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-methylpiperidin-2-one
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-({[4-(propan-2-yl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-(2-chlorophenyl)-2-hydroxy-1-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]ethan-1-one
5-ethanesulfonamido-1-methyl-2-phenyl-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
2-(5-{2-[methyl(1-methylpyrrolidin-3-yl)amino]ethyl}-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-1-yl)ethan-1-ol
2-[7-(oxan-4-yl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]pyridine-3-carbonitrile
3-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}methyl)-N-(pyridin-3-yl)benzamide
N-[(3R,4S)-1-(1-aminocyclopropanecarbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-6-(propan-2-yl)pyrimidin-4-amine
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
7-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-{5-[3-(3-fluoro-4-phenylbenzoyl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
3-(1-methylpiperidin-3-yl)-1-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]propan-1-one
3-{imidazo[1,2-a]pyridin-2-ylmethyl}-1-[4-(oxolan-2-ylmethoxy)phenyl]urea
1-[(3R,4R)-3-hydroxypiperidin-4-yl]-3-[2-(3-methylphenyl)-1,3-benzoxazol-6-yl]urea
4-(2-amino-5-ethylpyrimidin-4-yl)-N,N-dimethylpiperazine-1-sulfonamide
2-chloro-4-[1-(1-cyclopropylethyl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenol
2-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-4,6-dimethylpyridine-3-carbonitrile
1-cyclohexyl-4-{[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}piperazin-2-one
{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amine
(3aR,7aS)-2-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
5-{1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidin-4-yl}-5-(3-phenylpropyl)imidazolidine-2,4-dione
1-tert-butyl-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
3-(2-cyclohexylacetyl)-9-methoxy-N-methyl-7-oxo-N-(1,3-thiazol-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
ethyl 4-{[3-({1-[4-(3-fluorophenyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}piperazine-1-carboxylate
2-[2-fluoro-6-(propan-2-yloxy)phenyl]pyridine-4-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetamide
ethyl 3-({1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)-4-methylpentanoate