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N-[2-(2-methoxyethoxy)phenyl]-3-(pyridine-2-carbonyl)piperidine-1-carboxamide
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(pyridin-2-yl)ethan-1-one
4-(3-chlorophenoxy)-1-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
(2S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
3-[(dimethylamino)methyl]-1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-3-ol
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-ethyl-4-{[(4-fluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
2-(2-methoxyethyl)-1-[5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine
8-(2,2-dimethylpropyl)-1-(2-methoxyethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-3-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(dimethylamino)-N-{[1-(hydroxymethyl)cyclopentyl]methyl}-N-methyl-2-(2-methylphenyl)acetamide
N-{[7-chloro-2-(3-methylphenyl)quinolin-3-yl]methyl}-2-(2,5-dimethoxyphenyl)-N-(2-methoxyethyl)acetamide
2-[4-(2-methoxybenzoyl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
5-{[(2,3-dimethoxyphenyl)methyl]amino}-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
9-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-({2-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)pyridine-4-carboxamide
N-benzyl{[2-methyl-5-(6-oxo-1,6-dihydropyridazin-3-yl)phenyl]amino}sulfonamide
5-[(4-benzylpiperidin-1-yl)methyl]-N-(2-methylprop-2-en-1-yl)-1,2-oxazole-3-carboxamide
6,7-dimethoxy-3-[(2-methyl-1H-indol-5-yl)methyl]-3,4-dihydroquinazolin-4-one
3-[1-(1H-indol-5-yl)-1H-1,3-benzodiazol-2-yl]propan-1-ol
3-{1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]piperidin-3-yl}-N-[(3,4-difluorophenyl)methyl]propanamide
2-methoxy-1-(4-{4-[4-(methoxymethyl)piperidine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
N-methyl-5-oxo-1-phenyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-2,5-dihydro-1H-pyrazole-3-carboxamide
2-({[2-hydroxy-2-(4-hydroxyphenyl)ethyl]amino}methyl)-6-methylquinolin-4-ol
2-(4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-N-methyl-N-(2-phenylethyl)piperidin-3-amine
1-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-3-(1,2-oxazolidin-2-yl)propan-1-one
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]thiophene-2-carboxamide
5-{2-[2-(3-fluorophenyl)piperidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(2R,3R)-2-ethoxy-1'-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[4-(1H-pyrazol-1-yl)butan-2-yl]benzamide
2-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyridin-3-ol
[(2S)-1-{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl]methanol
N-[4-chloro-3-(3-propoxypiperidine-1-carbonyl)phenyl]acetamide
[1-(furan-3-carbonyl)-4-(2-phenylethyl)piperidin-4-yl]methanol
4-(2,3-dichlorophenyl)-1-[2-(pyrrolidin-1-yl)ethyl]-1H-1,2,3-triazole
1-(2-methylquinolin-6-yl)-3-[2-(pyrrolidin-1-yl)ethyl]urea
(3R,4R)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
3-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
1-methyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)piperidine-2-carboxamide
(3aR,5R,6S,7aS)-2-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-octahydro-1H-isoindole-5,6-diol
(2S,4S)-1-benzyl-N-ethyl-4-{[(3-hydroxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
N-{3-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-oxopropyl}methanesulfonamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-4,4,4-trifluoro-N-(oxolan-2-ylmethyl)butanamide
2-[4-(cyclopropylmethoxy)phenyl]-N,N-dimethylbenzamide
N-[(5-{[(3S)-3-ethylmorpholin-4-yl]methyl}furan-2-yl)methyl]-N-methylmethanesulfonamide
N-[1-(1H-indol-2-yl)ethyl]-N-methyl-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-(dicyclopropylmethyl)-N-methyl-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]acetamide
N-[2-(4-cyclopropyl-4H-1,2,4-triazol-3-yl)ethyl]aniline
(4aS,8aS)-4a-hydroxy-N-(1,3,4-thiadiazol-2-yl)-decahydroisoquinoline-2-carboxamide