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1-[2-(dimethyl-1,3-thiazol-4-yl)ethyl]-4-(3-fluorophenoxy)piperidine
(2S,4R)-4-{[(4-phenylphenyl)methyl]amino}-N-(propan-2-yl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-(1H-1,2,4-triazol-1-yl)propanamide
2-fluoro-6-(pyridin-3-yl)benzamide
[(2S)-1-{5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-2-yl]methanol
N-[1-(pyrazin-2-yl)propan-2-yl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
7-(2-methoxyethyl)-2-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(quinolin-8-yloxy)ethyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(5-methylpyrazin-2-yl)methyl]benzamide
7-(cyclohexylmethyl)-2-(oxan-4-yl)-2,7-diazaspiro[4.5]decane
6-{4-[1-(dimethylamino)ethyl]piperidin-1-yl}pyridine-2-carboxylic acid
(2R,3R,6R)-3-(2-methoxyphenyl)-5-[(1-methyl-1H-imidazol-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(1,3-thiazol-2-yl)-1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}piperidine
1-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-2-(pyridin-4-yl)ethan-1-one
4,4,4-trifluoro-1-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]butan-1-one
(4aS,7aR)-1-(2-cyclopropylacetyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-butyl-N-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-2,5-dihydro-1H-pyrrole-1-carboxamide
(7S,9aR)-N,7-dibenzyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-pyrazol-4-yl)ethyl]amine
N-[2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)propyl]-4-phenylbenzamide
N-{1-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
(1S,5R)-3-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(4-{4-[4-(2-hydroxyphenyl)piperazin-1-yl]piperidin-1-yl}phenyl)-N-(pyridin-2-ylmethyl)acetamide
N-[(2,4-dimethoxyphenyl)methyl]-5-(methoxymethyl)furan-2-carboxamide
5-[(1S,2R)-2-(butylcarbamoyl)cyclohexanecarbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(4-ethylphenyl)methyl]-N-methyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-ethyl-2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-4-carboxamide
8-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]benzamide
N,N-diethyl-1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
N-cyclopropyl-1-(furan-2-ylmethyl)-N-(3-phenylprop-2-yn-1-yl)piperidine-3-carboxamide
2-(benzyloxy)-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}ethan-1-one
9-methoxy-N-[(3-methoxyphenyl)methyl]-3-(3-methylbutyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-(2-{8-fluoro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-oxoethyl)-2,6-dimethyl-3,4-dihydropyrimidin-4-one
4-[2-(1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]morpholine
4-[2-hydroxy-2-(pyridin-3-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-(thiophen-2-ylmethyl)piperidine
N-[3-(3-fluorophenyl)phenyl]-1-[(6-methylpyridin-2-yl)methyl]piperidine-4-carboxamide
2-{4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
(1R,2R)-2-[({3-[2-(dimethylamino)ethoxy]phenyl}methyl)(ethyl)amino]cyclohexan-1-ol
7-(3-chlorophenyl)-4-(1-ethylpiperidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{2-methoxy-5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}morpholine
2-(2-methoxyethyl)-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1,3-benzoxazole-6-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(prop-2-en-1-yl)piperidin-3-amine
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]benzamide
(2S)-N-[2-(3,5-dimethylphenoxy)ethyl]-2-acetamido-N-methyl-4-(methylsulfanyl)butanamide
5-methyl-1-(4-methylphenyl)-4-[2-(pyridin-3-yl)acetyl]piperazin-2-one
N-methyl-1-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
5-{[butyl(furan-2-ylmethyl)amino]methyl}-N-(propan-2-yl)pyrimidin-2-amine
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1-methyl-1H-indole-2-carboxamide