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(1S,5R)-6-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[5-({[(2-chlorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
2-{1-[(2-methylphenyl)methyl]-4-(1,2-oxazol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
N-[2-(4-chlorophenyl)ethyl]-5-methyl-4-[(prop-2-en-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
1-(oxan-4-yl)-4-propanoyl-1,4-diazepane-6-carboxylic acid
1-[7-(1-hydroxy-2,2-diphenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-(thiophen-2-yl)butan-1-one
3-({cyclopropyl[(4-ethoxyphenyl)methyl]amino}methyl)-4H-chromen-4-one
[(3S,5S)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-3-yl]methanol
2-hydroxy-S-[3-(3-methoxypiperidine-1-carbonyl)phenyl]ethane-1-sulfonamido
9-[2-(2,6-dimethoxyphenoxy)ethyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
N-ethyl-2-(methoxymethyl)-4-oxo-1,3,8-triazaspiro[4.5]dec-1-ene-8-carboxamide
1-methyl-N-[2-(6-oxo-3-phenyl-1,4,5,6-tetrahydropyridazin-1-yl)ethyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
5-chloro-N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)thiophene-2-sulfonamide
3,5-dimethoxy-N-{[6-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
3-{1-[(2S)-1-acetylpyrrolidine-2-carbonyl]piperidin-4-yl}-N-[(4-fluorophenyl)methyl]propanamide
6-cyclopentyl-N-[(5,6-dimethylpyridin-3-yl)methyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-(thiophen-3-yl)propanamide
4-{[2-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
{3-[(2,4-difluorophenyl)methyl]-1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-3-yl}methanol
1-methyl-5-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
6-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
N-(2-hydroxyethyl)-5-(3-methylquinolin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-[3-({[5,8-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}amino)propyl]pyrrolidin-2-one
methyl 6-(but-3-enoyl)-2-[(cyclopropylmethyl)(propyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(4aR,7aS)-1-(1H-imidazol-4-ylmethyl)-4-(5-propyl-1,2-oxazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(2,6-difluorophenoxymethyl)-3-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1,2-oxazole
4-(4-fluoro-2-methylphenoxy)-1-[2-(methylamino)acetyl]piperidine-4-carboxylic acid
1-(2-methylpropyl)-5-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
3,5-dimethyl-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1,2-oxazole-4-carboxamide
5-(3-methoxyphenoxymethyl)-N-methyl-N-[4-(morpholin-4-yl)butyl]-1,2-oxazole-3-carboxamide
1-cyclopentyl-4-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazin-2-one
(1R,3S)-3-methoxy-7-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]-7-azaspiro[3.5]nonan-1-ol
N-[(6-chloropyridin-3-yl)methyl]-3-[(2-fluorophenyl)formamido]propanamide
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-5-methyl-1,2-oxazole-3-carboxamide
(3aR,6aR)-2-(3-chloro-4-methoxybenzoyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
3-({4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}methyl)benzonitrile
1-{3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidin-1-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)acetamide
N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-cyclobutyl-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-(4-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)-5-fluoropyrimidine
N-(2-fluoro-4-methylphenyl)-2-{[1-(morpholin-4-yl)propan-2-yl]amino}acetamide
3-{1-[3-(1H-indol-3-yl)propanoyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]benzamide
1-(4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}thiophen-2-yl)ethan-1-one
9-[(2R)-2-amino-2-phenylacetyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[1-(3,4-difluorobenzoyl)piperidin-4-yl]-2-phenylethyl}-N,1-dimethyl-1H-pyrazole-3-carboxamide
3-cyclopropyl-5-[2-(thiophen-2-yl)-1,3-thiazol-4-yl]-1H-1,2,4-triazole
3-hydroxy-3-{[4-(methoxymethyl)piperidin-1-yl]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one